SCHEMBL6309596

SCHEMBL6309596

Cc1ccccc1C1C2C(=O)N(Cc3ccccc3)C(=O)C2CN1C(=O)OCc1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CACNA1G O43497 1/20 0.43
CACNA1H O95180 1/20 0.43
CACNA1I Q9P0X4 1/20 0.43
CYP2D6 P10635 1/20 0.42
MAPK1 P28482 2/20 0.42
KMT2A Q03164 2/20 0.42
ALDH1A1 P00352 4/20 0.41
HTR2C P28335 1/20 0.41
MEN1 O00255 1/20 0.40
USP2 O75604 1/20 0.40
MAPT P10636 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
CASP1 P29466 1/20 0.40
CASP7 P55210 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5744862 0.89 CYP2D6 (0.41) CACNA1GCACNA1HCACNA1ICYP2D6ALDH1A1
SCHEMBL6319094 0.86 ALDH1A1 (0.45) CYP2D6MAPK1KMT2AALDH1A1HTR2C
SCHEMBL6310215 0.78 CACNA1G (0.44) CACNA1GCACNA1HCACNA1IHTR2C
SCHEMBL6310196 0.75 CACNA1G (0.44) CACNA1GCACNA1HCACNA1IHTR2C
SCHEMBL5747751 0.73 CACNA1G (0.43) CACNA1GCACNA1HCACNA1IHTR2C
SCHEMBL6310201 0.70 CACNA1G (0.44) CACNA1GCACNA1HCACNA1IHTR2C
SCHEMBL5745363 0.69 PARP1 (0.48)
SCHEMBL5517077 0.68 HTR2C (0.64) CACNA1GCACNA1HCACNA1IKMT2AALDH1A1
SCHEMBL5517082 0.68 HTR2C (0.64) CACNA1GCACNA1HCACNA1IKMT2AALDH1A1
SCHEMBL10053573 0.68 HTR2C (0.64) CACNA1GCACNA1HCACNA1IKMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050043354-A1 NK1 antagonist PFIZER INC 2005-02-24 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050043354-A1 NK1 antagonist TACR2, TACR1, TAC3 CACNA1G 1297/4885CACNA1H 1149/4885CACNA1I 1335/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.