SCHEMBL6312892

SCHEMBL6312892

CC1C(=O)[N]c2ccccc2-c2ccc(F)cc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 2/20 0.35
IDO1 P14902 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
MAPT P10636 1/20 0.33
SLC2A1 P11166 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ACHE P22303 1/20 0.33
GPR3 P46089 1/20 0.33
HTR7 P34969 1/20 0.32
HTR2B P41595 1/20 0.32
GSK3A P49840 2/20 0.32
GSK3B P49841 2/20 0.32
FLT3 P36888 1/20 0.32
CCNB2 O95067 1/20 0.32
CDK1 P06493 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6307251 0.88 ACHE (0.36) HSD11B1IDO1MEN1LMNAMAPT
SCHEMBL6306025 0.82 NOS3 (0.36) KMT2AACHEGPR3HTR7HTR2B
SCHEMBL12017094 0.76 HTR7 (0.45) HSD11B1MAPTMAPK1NPSR1GPR3
SCHEMBL5542657 0.71 NOS3 (0.40) MEN1MAPTKMT2A
SCHEMBL4415153 0.71 LRRK2 (0.41) IDO1MEN1KMT2AHTR7GSK3B
SCHEMBL4414735 0.69 IDO1 (0.37) IDO1MEN1KMT2AGPR3HTR7
Hydrochloric Acid SCHEMBL6306787 0.68 IDO1 (0.36) IDO1MEN1KMT2AGPR3HTR7
SCHEMBL6307367 0.66 HTR7 (0.34) IDO1HTR7HTR2B
SCHEMBL18634612 0.65 DAO (0.42) MEN1MAPTKMT2AFLT3
SCHEMBL8292982 0.64 GPR3 (0.41) GPR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6958330-B1 Polycyclic α-amino-ε-caprolactams and related compounds ELAN PHARMACEUTICALS, INC. (US) 2005-10-25 US claimed
EP-1042298-A1 POLYCYCLIC ALPHA-AMINO-EPSILON-CAPROLACTAMS AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2000-10-11 EP claimed
WO-1999032453-A1 POLYCYCLIC α-AMINO-⊂-CAPROLACTAMS AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 1999-07-01 WO claimed
US-6958330-B1 Polycyclic α-amino-ε-caprolactams and related compounds ELAN PHARMACEUTICALS, INC. (US) 2005-10-25 US disclosed
EP-1042298-A1 POLYCYCLIC ALPHA-AMINO-EPSILON-CAPROLACTAMS AND RELATED COMPOUNDS Elan Pharmaceuticals, Inc. (US) 2000-10-11 EP disclosed
WO-1999032453-A1 POLYCYCLIC α-AMINO-⊂-CAPROLACTAMS AND RELATED COMPOUNDS ELAN PHARMACEUTICALS, INC. (US) 1999-07-01 WO disclosed