SCHEMBL6315288

SCHEMBL6315288

Nc1ncc(-c2ccncc2)c(Nc2cnc3ccccc3c2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDGFRB P09619 1/20 0.49
PDGFRA P16234 1/20 0.49
ADORA2A P29274 1/20 0.48
ADORA1 P30542 1/20 0.48
ALDH1A1 P00352 2/20 0.46
NPC1 O15118 1/20 0.46
RAB9A P51151 1/20 0.46
GRM4 Q14833 1/20 0.46
TNF P01375 1/20 0.44
PIK3CA P42336 5/20 0.44
GSK3A P49840 1/20 0.43
GSK3B P49841 1/20 0.43
NPSR1 Q6W5P4 1/20 0.42
BUB1 O43683 1/20 0.42
FLT1 P17948 1/20 0.41
KDR P35968 1/20 0.41
KDM4E B2RXH2 1/20 0.40
PDE5A O76074 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6318945 0.87 TNF (0.44) ALDH1A1GRM4TNFPIK3CANPSR1
SCHEMBL6318862 0.85 DHFR (0.56) ADORA2AADORA1GRM4TNFPIK3CA
SCHEMBL6313731 0.84 PIK3CA (0.41) ADORA2AADORA1RAB9AGRM4TNF
SCHEMBL6312550 0.83 CA12 (0.56) ALDH1A1RAB9AGRM4TNFPIK3CA
SCHEMBL6320672 0.80 MAPT (0.50) RAB9APIK3CANPSR1SMN1; SMN2FAAH
SCHEMBL6313300 0.80 ABCG2 (0.46) ADORA2AADORA1GRM4TNFPIK3CA
SCHEMBL6312236 0.80 MAP4K4 (0.45) ADORA2AADORA1GRM4TNFPIK3CA
SCHEMBL6312017 0.79 CA2 (0.46) ALDH1A1RAB9ATNFPIK3CAKDM4E
SCHEMBL6313258 0.79 DYRK1A (0.43) ADORA2AADORA1GRM4TNFPIK3CA
SCHEMBL6312244 0.79 CYP1A2 (0.52) ADORA2AADORA1ALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6939874-B2 Substituted pyrimidinyl derivatives and methods of use AMGEN INC. (US) 2005-09-06 US disclosed