SCHEMBL632099

SCHEMBL632099

O=C(O)N1CCN(c2ccc(Cl)cc2)CC1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 4/20 0.68
ALDH1A1 P00352 2/20 0.68
AKR1C3 P42330 6/20 0.67
SMN1; SMN2 Q16637 3/20 0.67
HPGD P15428 1/20 0.67
HTT P42858 1/20 0.67
CHIA Q9BZP6 1/20 0.61
MEN1 O00255 2/20 0.59
KMT2A Q03164 2/20 0.59
HSP90AA1 P07900 1/20 0.59
MAPT P10636 2/20 0.59
GFER P55789 2/20 0.58
ATM Q13315 1/20 0.58
HTR1A P08908 1/20 0.57
HTR7 P34969 1/20 0.57
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
ME2 P23368 1/20 0.56
ME1 P48163 1/20 0.56
ME3 Q16798 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5233832 0.95 LMNA (0.62) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD
SCHEMBL1423584 0.85 AKR1C3 (0.67) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD
SCHEMBL28083212 0.83 AKR1C3 (0.65) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD
SCHEMBL3174172 0.83 CHIA (0.69) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD
SCHEMBL14276932 0.83 CASP6 (0.69) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD
SCHEMBL5414205 0.82 CHRM2 (0.52) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD
SCHEMBL3466014 0.82 TDP1 (0.64) LMNAALDH1A1SMN1; SMN2HTTMAPT
SCHEMBL631962 0.82 ALDH1A1 (0.69) LMNAALDH1A1AKR1C3HTTMEN1
SCHEMBL5231208 0.82 SRD5A2 (0.50) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD
SCHEMBL24158074 0.81 LMNA (0.85) LMNAALDH1A1AKR1C3SMN1; SMN2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234992-B1 PIPERAZINE DERIVATIVES AND THEIR USE AS LEPTIN RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2012-02-22 EP claimed
CN-102026975-A Piperazines as anti-obesity agents BIOVITRUM AB PUBL 2011-04-20 CN claimed
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed
CN-1602191-A Compounds and uses thereof for decreasing activity of hormone-sensitive lipase NOVO NORDISK AS (DK) 2005-03-30 CN claimed
US-20230121721-A1 MONOACYLGLYCEROL LIPASE INHIBITORS STICHTING HET NEDERLANDS KANKER INST ANTONI VAN LEEUWENHOEK ZIEKENHUIS (NL) 2023-04-20 US disclosed
EP-3875452-A1 MONOACYLGLYCEROL LIPASE INHIBITORS Stichting Het Nederlands Kanker Instituut- Antoni van Leeuwenhoek Ziekenhuis (NL) 2021-09-08 EP disclosed
EP-2473504-A2 HETEROCYCLIC COMPOUNDS FOR THE INHIBITION OF PASK Bioenergenix (US) 2012-07-11 EP disclosed
CN-102026975-A Piperazines as anti-obesity agents BIOVITRUM AB PUBL 2011-04-20 CN disclosed
CN-102015668-A Piperazine derivatives and their use as leptin receptor modulators ASTRAZENECA AB PUBL 2011-04-13 CN disclosed
WO-2011028947-A2 HETEROCYCLIC COMPOUNDS FOR THE INHIBITION OF PASK BIOENERGENIX (US) 2011-03-10 WO disclosed
US-20080261956-A1 Substituted Phenols as Active Agents Inhibiting Vegf Production PTC THERAPEUTICS, INC. 2008-10-23 US disclosed
CN-1326519-C Compounds and uses thereof for decreasing activity of hormone-sensitive lipase NOVO NORDISK AS (DK) 2007-07-18 CN disclosed
CN-1602191-A Compounds and uses thereof for decreasing activity of hormone-sensitive lipase NOVO NORDISK AS (DK) 2005-03-30 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230121721-A1 MONOACYLGLYCEROL LIPASE INHIBITORS MGLL, PNLIP, LIPA LMNA 926/4885ALDH1A1 932/4885AKR1C3 1792/4885
US-20080261956-A1 Substituted Phenols as Active Agents Inhibiting Vegf Production VEGFA, FLT4, FLT1 LMNA 4326/4885ALDH1A1 936/4885AKR1C3 1425/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.