SCHEMBL6324748

SCHEMBL6324748

O=C(Cl)c1cc(F)c(F)c(F)c1O

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
ALOX15 P16050 1/20 0.43
CES2 O00748 3/20 0.39
CES1 P23141 3/20 0.39
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA4 P22748 2/20 0.35
HSD17B1 P14061 9/20 0.35
HSD17B2 P37059 9/20 0.35
KEAP1 Q14145 1/20 0.34
NFE2L2 Q16236 1/20 0.34
POLB P06746 1/20 0.34
APEX1 P27695 1/20 0.34
PIK3CA P42336 1/20 0.33
ALB P02768 1/20 0.32
ERN1 O75460 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7813170 0.84 HSD17B1 (0.45) ALDH1A1ALOX15CES2CES1HSD17B1
SCHEMBL345016 0.84 ALDH1A1 (0.48) ALDH1A1ALOX15CES2CES1CA1
SCHEMBL6324251 0.80 AKR1C2 (0.48) ALDH1A1CES2CES1CA1CA2
SCHEMBL155657 0.78 KMT2A (0.41) ALDH1A1CES2CES1CA1CA2
SCHEMBL8072641 0.78 ALDH1A1 (0.43) ALDH1A1ALOX15CES2CES1CA1
SCHEMBL1408469 0.77 ALDH1A1 (0.42) ALDH1A1ALOX15CES2CES1CA1
SCHEMBL24710385 0.76 ALDH1A1 (0.54) ALDH1A1ALOX15CES2CES1CA1
SCHEMBL28525271 0.76 ALDH1A1 (0.54) ALDH1A1ALOX15CES2CES1CA1
SCHEMBL8160121 0.76 ALDH1A1 (0.45) ALDH1A1ALOX15CES2CES1CA1
SCHEMBL29690316 0.76 ALDH1A1 (0.45) ALDH1A1ALOX15CES2CES1CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050124664-A1 Urea thiadiazole inhibitors of plasminogen activator inhibior-1 BRISTOL-MYERS SQUIBB CO. 2005-06-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050124664-A1 Urea thiadiazole inhibitors of plasminogen activator inhibior-1 SERPINE1, SERPINC1, SERPINB1 ALDH1A1 155/4885ALOX15 1940/4885CES2 3089/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.