SCHEMBL6326207

SCHEMBL6326207

O=C(CS(=O)(=O)N1CCOCC1)c1ccc([N+](=O)[O-])o1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.59
DDIT3 P35638 8/20 0.57
RAB9A P51151 4/20 0.57
MAPT P10636 3/20 0.57
KMT2A Q03164 2/20 0.57
MITF O75030 3/20 0.51
SMN1; SMN2 Q16637 2/20 0.51
NPC1 O15118 2/20 0.50
THRB P10828 1/20 0.48
CSF1R P07333 1/20 0.47
HSP90AA1 P07900 1/20 0.47
POLB P06746 3/20 0.45
GAA P10253 2/20 0.45
MEN1 O00255 1/20 0.45
HTT P42858 1/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
CA9 Q16790 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5322339 0.74 ALDH1A1 (1.00) ALDH1A1DDIT3RAB9AMAPTKMT2A
SCHEMBL16919773 0.73 DDIT3 (1.00) ALDH1A1DDIT3RAB9AMAPTKMT2A
SCHEMBL8896530 0.70 ALDH1A1 (0.58) ALDH1A1MAPTKMT2ASMN1; SMN2MEN1
SCHEMBL11455980 0.70 LMNA (0.56) ALDH1A1RAB9AMAPTKMT2AMITF
SCHEMBL12261479 0.70 LMNA (0.53) ALDH1A1RAB9AMAPTKMT2AMITF
SCHEMBL6427316 0.69 RAB9A (0.74) ALDH1A1DDIT3RAB9AMAPTKMT2A
SCHEMBL6203436 0.69 ATM (0.46) ALDH1A1MAPTKMT2ANPC1GAA
SCHEMBL11790220 0.69 LMNA (0.51) ALDH1A1RAB9AMAPTKMT2AMITF
Nifurmerone SCHEMBL398798 0.69 LMNA (0.51) ALDH1A1RAB9AMAPTKMT2AMITF
SCHEMBL4186870 0.69 LMNA (0.65) ALDH1A1MAPTKMT2ASMN1; SMN2GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1501830-A1 7-ARYL-3,9-DIAZABICYCLO[3.3.1]NON-6-ENE DERIVATIVES AND THEIR USE AS RENIN INHIBITORS IN THE TREATMENT OF HYPERTENSION, CARDIOVASCULAR OR RENAL DISEASES Actelion Pharmaceuticals Ltd. (CH) 2005-02-02 EP claimed
WO-2003093267-A1 7-ARYL-3,9-DIAZABICYCLO(3.3.1)NON-6-ENE DERIVATIVES AND THEIR USE AS RENIN INHIBITORS IN THE TREATMENT OF HYPERTENSION, CARDIOVASCULAR OR RENAL DISEASES ACTELION PHARMACEUTICALS LTD (CH) 2003-11-13 WO claimed
US-20050272036-A1 Ketones ASTRAZENECA AB (SE) 2005-12-08 US disclosed