SCHEMBL6330560

SCHEMBL6330560

CN(C)Cc1cn(S(=O)(=O)c2ccc3c(c2)CNCC3(C)C)c2ccccc12

nearest known ligand 0.58

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 17/20 0.58
HDAC1 Q13547 2/20 0.52
HDAC2 Q92769 2/20 0.52
HDAC6 Q9UBN7 2/20 0.52
HTR1A P08908 1/20 0.46
DRD2 P14416 1/20 0.46
HTR1D P28221 1/20 0.46
HTR1B P28222 1/20 0.46
HTR1F P30939 1/20 0.46
HTR7 P34969 1/20 0.46
DRD3 P35462 1/20 0.46
TNFSF11 O14788 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6331024 0.85 HTR6 (0.52) HTR6
SCHEMBL6335588 0.84 HTR6 (0.60) HTR6HDAC1HDAC2HDAC6HTR1A
SCHEMBL6166554 0.82 HTR6 (0.63) HTR6HDAC1HDAC2HDAC6HTR1A
SCHEMBL1171841 0.75 HTR6 (1.00) HTR6HDAC1HDAC2HDAC6HTR1A
SCHEMBL3248158 0.73 HTR6 (1.00) HTR6HDAC1HDAC2HDAC6HTR1A
SCHEMBL6404989 0.72 HTR6 (0.54) HTR6
SCHEMBL6336170 0.69 PNMT (0.50) HTR6
SCHEMBL6332940 0.68 HTR6 (0.51) HTR6HTR1ADRD2
SCHEMBL6328502 0.68 HTR6 (0.40) HTR6HTR1ADRD2
SCHEMBL949155 0.67 HTR6 (0.65) HTR6HDAC1HDAC2HDAC6HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849644-B2 Isoquinoline derivatives useful in the treatment of CNS disorders SMITHKLINE BEECHAM P.L.C. (GB) 2005-02-01 US claimed