SCHEMBL6333359

SCHEMBL6333359

Fc1cc(Br)c2ccoc2c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.34
ALDH1A1 P00352 3/20 0.33
CYP3A4 P08684 2/20 0.33
CYP2A6 P11509 2/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAOA P21397 2/20 0.33
MAOB P27338 1/20 0.33
FTO Q9C0B1 1/20 0.32
KCNA3 P22001 3/20 0.32
KCNA5 P22460 2/20 0.32
KDM4E B2RXH2 2/20 0.31
CYP1A1 P04798 1/20 0.31
CYP1A2 P05177 1/20 0.31
PGR P06401 1/20 0.31
ADORA3 P0DMS8 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2C9 P11712 1/20 0.31
KCNA2 P16389 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16432225 0.78 CYP3A4 (0.35) ALDH1A1CYP3A4CYP2A6MAPTHPGD
SCHEMBL26540300 0.78 TRPA1 (0.42) TRPA1ALDH1A1CYP3A4CYP2A6MAPT
SCHEMBL806507 0.75 TRPA1 (0.37) TRPA1ALDH1A1CYP3A4CYP2A6MAPT
SCHEMBL20839528 0.75 CYP3A4 (0.34) ALDH1A1CYP3A4CYP2A6MAPTHPGD
SCHEMBL28859634 0.75 MAOA (0.37) ALDH1A1CYP3A4CYP2A6MAPTHPGD
SCHEMBL23330372 0.71 CYP11B1 (0.42) ALDH1A1HPGDMAOAMAOBKDM4E
SCHEMBL29144468 0.71 FTO (0.41) ALDH1A1CYP3A4CYP2A6MAPTHPGD
SCHEMBL6334853 0.71 TRPA1 (0.34) TRPA1ALDH1A1CYP3A4CYP2A6MAPT
SCHEMBL16048354 0.68 MAOA (0.36) TRPA1MAOAMAOBFTOIDO1
SCHEMBL4351751 0.68 ALDH1A1 (0.37) TRPA1ALDH1A1CYP3A4CYP2A6L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6881733-B1 Serotonergic benzofurans ELI LILLY AND COMPANY (US) 2005-04-19 US disclosed
EP-1204659-B1 SEROTONERGIC BENZOFURANS LILLY CO ELI (US) 2003-11-26 EP disclosed
EP-1204659-A2 SEROTONERGIC BENZOFURANS ELI LILLY AND COMPANY (US) 2002-05-15 EP disclosed
WO-2001009122-A2 SEROTONERGIC BENZOFURANS ELI LILLY AND COMPANY (US) 2001-02-08 WO disclosed