SCHEMBL633558

SCHEMBL633558

CC1=C(C)C2=C(CCC(C)(C)O2)C(=O)C1=O

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MALT1 Q9UDY8 9/20 0.58
IDO1 P14902 2/20 0.58
KDM4E B2RXH2 1/20 0.58
MEN1 O00255 1/20 0.58
CES2 O00748 1/20 0.58
GMNN O75496 1/20 0.58
TDP2 O95551 1/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
TP53 P04637 1/20 0.58
CYP1A2 P05177 1/20 0.58
GLA P06280 1/20 0.58
CYP3A4 P08684 1/20 0.58
CYP2D6 P10635 1/20 0.58
MAPT P10636 1/20 0.58
HSPD1 P10809 1/20 0.58
THRB P10828 1/20 0.58
CYP2C9 P11712 1/20 0.58
NQO1 P15559 1/20 0.58
ALOX15 P16050 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13052458 0.84 IDO1 (0.47) MALT1IDO1KDM4EMEN1CES2
SCHEMBL5940394 0.74 MALT1 (0.74) MALT1IDO1KDM4EMEN1CES2
SCHEMBL12140550 0.74 MALT1 (0.55) MALT1IDO1KDM4EMEN1CES2
Lapachone SCHEMBL107042 0.74 MALT1 (1.00) MALT1IDO1KDM4EMEN1CES2
Alpha-Lapachone SCHEMBL102553 0.72 IDO1 (1.00) MALT1IDO1KDM4EMEN1CES2
SCHEMBL5940435 0.71 MALT1 (0.75) MALT1IDO1KDM4EMEN1CES2
SCHEMBL14439372 0.69 MALT1 (0.90) MALT1IDO1KDM4EMEN1CES2
SCHEMBL14456608 0.69 MALT1 (0.71) MALT1IDO1KDM4EMEN1CES2
SCHEMBL5940140 0.69 MALT1 (0.71) MALT1IDO1KDM4EMEN1CES2
SCHEMBL8186444 0.67 MALT1 (0.76) MALT1IDO1KDM4EMEN1CES2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012153162-A1 NOVEL METHOD FOR PREPARATION OF ATOVAQUONE LUPIN LIMITED (IN) 2012-11-15 WO disclosed
EP-2419095-A2 PHARMACEUTICALLY ACTIVE COMPOSITIONS COMPRISING OXIDATIVE STRESS MODULATORS (OSM), NEW CHEMICAL ENTITIES, COMPOSITIONS AND USES Colby Pharmaceutical Company (US) 2012-02-22 EP disclosed
US-20100297262-A1 PHARMACEUTICALLY ACTIVE COMPOSITIONS COMPRISING OXIDATIVE STRESS MODULATORS (OSM), NEW CHEMICAL ENTITIES, COMPOSITIONS AND USES COLBY PHARMACEUTICAL COMPANY (US) 2010-11-25 US disclosed
US-20100297262-A1 PHARMACEUTICALLY ACTIVE COMPOSITIONS COMPRISING OXIDATIVE STRESS MODULATORS (OSM), NEW CHEMICAL ENTITIES, COMPOSITIONS AND USES COLBY PHARMACEUTICAL COMPANY (US) 2010-11-25 US disclosed
US-20100297262-A1 PHARMACEUTICALLY ACTIVE COMPOSITIONS COMPRISING OXIDATIVE STRESS MODULATORS (OSM), NEW CHEMICAL ENTITIES, COMPOSITIONS AND USES COLBY PHARMACEUTICAL COMPANY (US) 2010-11-25 US disclosed
WO-2010121177-A2 PHARMACEUTICALLY ACTIVE COMPOSITIONS COMPRISING OXIDATIVE STRESS MODULATORS (OSM), NEW CHEMICAL ENTITIES, COMPOSITIONS AND USES COLBY PHARMACEUTICAL COMPANY (US) 2010-10-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100297262-A1 PHARMACEUTICALLY ACTIVE COMPOSITIONS COMPRISING OXIDATIVE STRESS MODULATORS (OSM), NEW CHEMICAL ENTITIES, COMPOSITIONS AND USES MPO, HMOX1, LPO MALT1 2646/4885IDO1 838/4885KDM4E 4586/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.