SCHEMBL6352535

SCHEMBL6352535

CCOCCN1CCC(C(=O)OC(C)(C)C)=Cc2cc(Br)ccc21

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 3/20 0.36
GABRG2 P18507 3/20 0.36
GABRB3 P28472 3/20 0.36
GABRA5 P31644 3/20 0.36
GABRA3 P34903 3/20 0.36
GABRA2 P47869 3/20 0.36
GABRA6 Q16445 3/20 0.36
GABRB2 P47870 1/20 0.36
GABRA4 P48169 1/20 0.33
SRD5A1 P18405 1/20 0.32
RBP4 P02753 1/20 0.32
KMT2A Q03164 3/20 0.32
ALDH1A1 P00352 2/20 0.32
PKM P14618 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HRH2 P25021 1/20 0.32
GPR119 Q8TDV5 1/20 0.32
MEN1 O00255 2/20 0.31
BACE1 P56817 1/20 0.30
WDR5 P61964 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6343396 0.90 GABRA1 (0.37) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6343215 0.90 GABRA1 (0.38) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6352550 0.86 HRH2 (0.39) KMT2AALDH1A1HRH2MEN1WDR5
SCHEMBL5206682 0.82 GABRA1 (0.43) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7547077 0.79 ALDH1A1 (0.40) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL7541560 0.78 ALDH1A1 (0.36) KMT2AALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL7540580 0.77 GABRG2 (0.38) GABRA1GABRG2GABRB3GABRA5GABRA3
SCHEMBL6339852 0.76 ALDH1A1 (0.38) KMT2AALDH1A1SMN1; SMN2MEN1LMNA
SCHEMBL6341635 0.75 SMN1; SMN2 (0.35) KMT2AALDH1A1SMN1; SMN2MEN1POLB
SCHEMBL6350680 0.74 LMNA (0.40) RBP4KMT2AALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6936602-B1 Benzazepine derivatives, process for the preparation of the same and uses thereof TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2005-08-30 US disclosed
EP-1186604-A1 BENZAZEPINE DERIVATIVES, PROCESS FOR THE PREPARATION OF THE SAME AND USES THEREOF Takeda Chemical Industries, Ltd. (JP) 2002-03-13 EP disclosed