SCHEMBL6354855

SCHEMBL6354855

O=C1C=CC(=O)N1c1cn(Cc2cccc3ccccc23)c2ccccc12

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.48
ALDH1A1 P00352 4/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
KMT2A Q03164 2/20 0.48
MEN1 O00255 1/20 0.48
APAF1 O14727 1/20 0.48
CYP1A2 P05177 1/20 0.48
GAA P10253 1/20 0.48
THRB P10828 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
BLM P54132 1/20 0.48
KDM4C Q9H3R0 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
PTPN1 P18031 1/20 0.47
KDM4E B2RXH2 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HTT P42858 2/20 0.45
MCL1 Q07820 4/20 0.44
BAD Q92934 4/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6352429 0.77 AKR1B1 (0.43) L3MBTL1CYP1A2SMN1; SMN2CHRM1LMNA
SCHEMBL6353710 0.77 MGLL (0.50) MAPTALDH1A1KMT2AMEN1MGLL
SCHEMBL6346957 0.74 MEN1 (0.48) MAPTALDH1A1KMT2AMEN1GAA
SCHEMBL5410439 0.74 CNR2 (0.47) MGLLCHRM1CNR2
SCHEMBL6802017 0.73 ALDH1A1 (0.55) MAPTALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL6802019 0.73 ALDH1A1 (0.70) MAPTALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL718459 0.73 PTGS1 (0.58) MAPTALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL21999706 0.72 LMNA (0.69) MCL1BADCHRM1LMNACNR2
SCHEMBL8758329 0.70 HTR2A (0.53) MAPTALDH1A1L3MBTL1KMT2AMEN1
SCHEMBL152339 0.70 TLR9 (0.64) MAPTALDH1A1TDP1MGLLPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6849643-B2 Indazolyl-substituted pyrroline compounds as kinase inhibitors ORTHO-MCNEIL PHARMACEUTICAL, INC. (US) 2005-02-01 US disclosed