SCHEMBL635858

SCHEMBL635858

CC(C)(C)NC(=O)N[C@H](C(=O)O)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.39
CA2 P00918 1/20 0.39
POLB P06746 1/20 0.38
NPC1 O15118 3/20 0.37
RAB9A P51151 3/20 0.37
MAPT P10636 1/20 0.37
ELANE P08246 2/20 0.34
MMP2 P08253 4/20 0.33
MMP3 P08254 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
EPHX2 P34913 1/20 0.32
PYGL P06737 1/20 0.32
CYP2C9 P11712 1/20 0.32
PDF Q9HBH1 1/20 0.31
HDAC4 P56524 1/20 0.31
HDAC1 Q13547 1/20 0.31
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL635859 1.00 TRPA1 (0.39) TRPA1CA2POLBNPC1RAB9A
SCHEMBL4372546 1.00 TRPA1 (0.39) TRPA1CA2POLBNPC1RAB9A
SCHEMBL14943545 0.83 TRPA1 (0.39) TRPA1POLBNPC1RAB9AMAPT
SCHEMBL12401122 0.81 TRPA1 (0.38) TRPA1POLBNPC1RAB9AMAPT
SCHEMBL636880 0.79 TRPA1 (0.37) TRPA1POLBNPC1RAB9AMAPT
SCHEMBL636879 0.79 TRPA1 (0.37) TRPA1POLBNPC1RAB9AMAPT
SCHEMBL12571864 0.78 TRPA1 (0.36) TRPA1POLBNPC1RAB9AMAPT
SCHEMBL12482473 0.78 TRPA1 (0.36) TRPA1POLBNPC1RAB9AMAPT
SCHEMBL10107206 0.78 CTSK (0.37) TRPA1CA2POLBNPC1RAB9A
SCHEMBL13135688 0.77 TRPA1 (0.53) TRPA1POLBMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 87 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2014061034-A1 PROCESS FOR PREPARATION OF BOCEPREVIR AND INTERMEDIATES THEREOF MSN LABORATORIES LIMITED (IN) 2014-04-24 WO claimed
US-20230212116-A1 SARS-COV-2 MAIN PROTEASE INHIBITORS THE TEXAS A&M UNIVERSITY SYSTEM 2023-07-06 US disclosed
EP-2528922-B1 POLYHETEROCYCLIC COMPOUNDS AS HCV INHIBITORS AB PHARMA LTD (CN) 2017-08-02 EP disclosed
EP-1906945-B1 HCV INHIBITORS VIROBAY INC (US) 2015-08-05 EP disclosed
CN-103396344-B One-pot synthetic method for N-t-butyl-aminocarbonyl-3-methyl-L-valine SUZHOU UUGENE BIOPHARMA CO., LTD. (CN) 2014-10-29 CN disclosed
CN-103396344-B One-pot synthetic method for N-t-butyl-aminocarbonyl-3-methyl-L-valine SUZHOU UUGENE BIOPHARMA CO., LTD. (CN) 2014-10-29 CN disclosed
WO-2014061034-A1 PROCESS FOR PREPARATION OF BOCEPREVIR AND INTERMEDIATES THEREOF MSN LABORATORIES LIMITED (IN) 2014-04-24 WO disclosed
WO-2013178682-A2 MULTICOMPONENT PROCESS FOR THE PREPARATION OF BICYCLIC COMPOUNDS CHEMO IBÉRICA, S.A. (ES) 2013-12-05 WO disclosed
CN-103396344-A One-pot synthetic method for N-t-butyl-aminocarbonyl-3-methyl-L-valine SUZHOU UUGENE BIOPHARMA CO LTD 2013-11-20 CN disclosed
CN-103396344-A One-pot synthetic method for N-t-butyl-aminocarbonyl-3-methyl-L-valine SUZHOU UUGENE BIOPHARMA CO LTD 2013-11-20 CN disclosed
US-20070265281-A1 Organic Compounds and Their Uses COTTENS SYLVAIN 2007-11-15 US disclosed
WO-2007121124-A2 HCV INHIBITORS COMPRISING BETA AMINO ACIDS AND THEIR USES NOVARTIS AG (CH) 2007-10-25 WO disclosed
WO-2007121125-A2 HCV INHIBITORS NOVARTIS AG (CH) 2007-10-25 WO disclosed
US-20070243166-A1 Hepatitis C Inhibitor Compounds LLINAS-BRUNET MONTSE 2007-10-18 US disclosed
US-20070243166-A1 Hepatitis C Inhibitor Compounds LLINAS-BRUNET MONTSE 2007-10-18 US disclosed
US-20070054864-A1 1-[2S-(3-Tert-butylureido)-3,3-dimethylbutyryl]-4R-(7-methoxy-2-pyrazol-1-yl-quinolin-4-yloxy)-pyrrolidine-2S-carboxylic acid (1S-cyclopropylaminooxalylbutyl)amide, for example; useful in treating hepatitis C infections QUEST DIAGNOSTICS INVESTMENTS LLC 2007-03-08 US disclosed
US-20070054864-A1 1-[2S-(3-Tert-butylureido)-3,3-dimethylbutyryl]-4R-(7-methoxy-2-pyrazol-1-yl-quinolin-4-yloxy)-pyrrolidine-2S-carboxylic acid (1S-cyclopropylaminooxalylbutyl)amide, for example; useful in treating hepatitis C infections QUEST DIAGNOSTICS INVESTMENTS LLC 2007-03-08 US disclosed
US-20070054864-A1 1-[2S-(3-Tert-butylureido)-3,3-dimethylbutyryl]-4R-(7-methoxy-2-pyrazol-1-yl-quinolin-4-yloxy)-pyrrolidine-2S-carboxylic acid (1S-cyclopropylaminooxalylbutyl)amide, for example; useful in treating hepatitis C infections QUEST DIAGNOSTICS INVESTMENTS LLC 2007-03-08 US disclosed
WO-2007005838-A2 HCV INHIBITORS VIROBAY, INC. (US) 2007-01-11 WO disclosed
WO-2007005838-A2 HCV INHIBITORS VIROBAY, INC. (US) 2007-01-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230212116-A1 SARS-COV-2 MAIN PROTEASE INHIBITORS ACE2, ACE, TMPRSS2 TRPA1 2898/4885CA2 964/4885POLB 676/4885
US-20070243166-A1 Hepatitis C Inhibitor Compounds HAVCR2, CTRL, CTRC TRPA1 3947/4885CA2 4311/4885POLB 3280/4885
US-20070054864-A1 1-[2S-(3-Tert-butylureido)-3,3-dimethylbutyryl]-4R-(7-methoxy-2-pyrazol-1-yl-quinolin-4-yloxy)-pyrrolidine-2S-carboxylic acid (1S-cyclopropylaminooxalylbutyl)amide, for example; useful in treating hepatitis C infections HAVCR2, EIF2AK2, GTF3C1 TRPA1 4504/4885CA2 4790/4885POLB 263/4885
US-20070265281-A1 Organic Compounds and Their Uses OAT, OTC, AOX1 TRPA1 748/4885CA2 1716/4885POLB 419/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.