SCHEMBL6364443

SCHEMBL6364443

COc1ccc2cccc(N3CCN(CCNC(=O)c4ccc(F)cc4)CC3)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 1.00
KDM4E B2RXH2 1/20 1.00
ALDH1A1 P00352 1/20 1.00
CYP1A2 P05177 1/20 1.00
CYP3A4 P08684 1/20 1.00
MAPT P10636 1/20 1.00
HPGD P15428 1/20 1.00
MAPK1 P28482 1/20 1.00
HSD17B10 Q99714 1/20 1.00
DRD4 P21917 9/20 0.70
DRD2 P14416 7/20 0.68
ADRA2A P08913 2/20 0.65
ADRA1D P25100 1/20 0.59
ADRA1A P35348 1/20 0.59
ADRA1B P35368 1/20 0.59
DRD3 P35462 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3187184 0.99 HTR1A (0.98) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9843330 0.94 HTR1A (0.88) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9640147 0.93 HTR1A (0.87) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9280229 0.93 HTR1A (0.86) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9639153 0.92 HTR1A (0.85) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9198697 0.87 HTR1A (0.76) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9639119 0.86 HTR1A (0.75) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9282819 0.85 HTR1A (0.73) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
SCHEMBL9843542 0.84 HTR1A (0.73) HTR1AKDM4EALDH1A1CYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9640094 0.84 HTR1A (0.72) HTR1AKDM4EALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US claimed
EP-0434561-B1 1-Naphthyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-10-18 EP claimed
US-5143916-A Hypotensive agents ADIR ET COMPAGNIE (FR) 1992-09-01 US claimed
EP-0434561-A2 1-Naphthyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-06-26 EP claimed
JP-3291275-A None JP disclosed
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS INC (US) 2025-09-25 US disclosed
US-20230414628-A1 METHODS FOR TREATING DISEASES MEDIATED BY GLUTATHIONE PEROXIDASE 4 RAMESH SANATH KUMAR (US) 2023-12-28 US disclosed
WO-2023212244-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS TESSELLATE THERAPEUTICS, INC. (US) 2023-11-02 WO disclosed
US-20220244263-A1 METHODS FOR TREATING SMALL CELL NEUROENDOCRINE AND RELATED CANCERS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2022-08-04 US disclosed
US-20050004105-A1 Treatment for a attention-deficit hyperactivity disorder PSYCHOGENCIS, INC. 2005-01-06 US disclosed
EP-1067965-B1 PHARMACEUTICAL COMPOSITION FOR TREATING CEREBRAL APOPLEXY AND CRANIOCEREBRAL TRAUMA BAYER HEALTHCARE AG (DE) 2004-09-29 EP disclosed
WO-2004069339-A1 TREATMENT FOR ATTENTION-DEFICIT HYPERACTIVITY DISORDER PSYCHOGENICS INC. (US) 2004-08-19 WO disclosed
EP-1067965-A1 PHARMACEUTICAL COMPOSITION FOR TREATING CEREBRAL APOPLEXY AND CRANIOCEREBRAL TRAUMA Bayer Aktiengesellschaft (DE) 2001-01-17 EP disclosed
EP-0969842-A1 PHARMACEUTICAL COMPOSITION R.P. Scherer Limited (GB) 2000-01-12 EP disclosed
WO-1999029346-A1 PHARMACEUTICAL COMPOSITION FOR TREATING CEREBRAL APOPLEXY AND CRANIOCEREBRAL TRAUMA BAYER AKTIENGESELLSCHAFT (DE) 1999-06-17 WO disclosed
WO-1998042344-A1 PHARMACEUTICAL COMPOSITION R. P. SCHERER LIMITED (GB) 1998-10-01 WO disclosed
EP-0434561-B1 1-Naphthyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 1995-10-18 EP disclosed
US-5166157-A Analgesics, antidepressants or psychological disorders ADIR ET COMPAGNIE (FR) 1992-11-24 US disclosed
JP-H03291275-A NEW (1-NAPHTHYL)PIPERAZINE DERIVATIVE, PREPARATION OF THE SAME, AND COMPOSITION OF DRUG INCLUDING THE SAME ADIR 1991-12-20 JP disclosed
EP-0434561-A2 1-Naphthyl-piperazine derivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1991-06-26 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004105-A1 Treatment for a attention-deficit hyperactivity disorder HTR1A, HTR5A, HTR2A HTR1A 1/4885KDM4E 3338/4885ALDH1A1 351/4885
US-20250295611-A1 METHODS OF TREATING 5HT2A RECEPTOR-MEDIATED CONDITIONS HTR2A, HTR5A, HTR6 HTR1A 4/4885KDM4E 4347/4885ALDH1A1 913/4885
US-20230414628-A1 METHODS FOR TREATING DISEASES MEDIATED BY GLUTATHIONE PEROXIDASE 4 GPX4, GPX1, MPO HTR1A 3582/4885KDM4E 3107/4885ALDH1A1 493/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.