SCHEMBL6375010

SCHEMBL6375010

CC[C@H](C)[C@@H](N)C(=O)NCC(C)Cc1cccc(N(CC(C)C)S(=O)(=O)c2ccccc2)c1O

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.39
BCL2L1 Q07817 3/20 0.39
RORC P51449 5/20 0.38
GPR88 Q9GZN0 4/20 0.35
MMP2 P08253 1/20 0.35
LARS1 Q9P2J5 1/20 0.34
HPGD P15428 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL5506705 0.86 KEAP1 (0.38) RORCMMP2HPGD
SCHEMBL5029070 0.84 MMP2 (0.43) RORCMMP2HPGD
SCHEMBL7458622 0.80 RORC (0.45) MCL1BCL2L1RORCHPGD
SCHEMBL5981554 0.79 MCL1 (0.39) MCL1BCL2L1HPGD
SCHEMBL4854967 0.78 ESR1 (0.44)
SCHEMBL7455250 0.75 ADAM17 (0.37) MCL1BCL2L1MMP2HPGD
SCHEMBL5691126 0.74 KEAP1 (0.39) RORCMMP2HPGD
Hydrochloric Acid SCHEMBL6394136 0.74 KEAP1 (0.35) MCL1RORCMMP2
SCHEMBL6390909 0.73 HSD11B1 (0.37) RORCMMP2HPGD
SCHEMBL4853866 0.73 RORC (0.44) MCL1BCL2L1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0813543-B1 BIS-AMINO ACID HYDROXYETHYLAMINO SULFONAMIDE RETROVIRAL PROTEASE INHIBITORS SEARLE LLC (US) 2005-09-14 EP disclosed
EP-1076062-A1 Bis-amino acid hydroxyethylamino sulfonamide retroviral protease inhibitors G.D. SEARLE & CO. (US) 2001-02-14 EP disclosed