SCHEMBL6375427

SCHEMBL6375427

COc1ccccc1CNC(Cc1ccccc1)C(=O)O

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.73
ITGB7 P26010 1/20 0.73
ALDH1A1 P00352 3/20 0.73
GAA P10253 1/20 0.73
MEN1 O00255 2/20 0.57
KMT2A Q03164 2/20 0.57
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
ATM Q13315 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HPGD P15428 2/20 0.52
HTT P42858 2/20 0.51
TAAR1 Q96RJ0 1/20 0.51
FPR2 P25090 1/20 0.51
BCHE P06276 3/20 0.51
LMNA P02545 1/20 0.50
BACE1 P56817 1/20 0.49
ALOX15 P16050 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6375429 1.00 ITGA4 (0.73) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL3857463 0.86 ITGA4 (0.57) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL3857454 0.86 ITGA4 (0.57) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL30340352 0.86 PDCD1 (0.61) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL7390734 0.84 ALDH1A1 (0.67) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL5215651 0.84 ALDH1A1 (0.67) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL5215743 0.80 ALDH1A1 (0.61) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL2247336 0.80 ITGA4 (0.53) ITGA4ITGB7ALDH1A1GAAMEN1
SCHEMBL28047718 0.80 PTPN1 (0.61) ITGA4ITGB7ALDH1A1GAAKMT2A
SCHEMBL28047720 0.80 PTPN1 (0.61) ITGA4ITGB7ALDH1A1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1001764-A4 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO INC (US) 2005-08-24 EP disclosed
US-6903075-B1 Heterocyclic amide compounds as cell adhesion inhibitors MERCK & CO., INC. (US) 2005-06-07 US disclosed
EP-1001764-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS Merck & Co., Inc. (a New Jersey corp.) (US) 2000-05-24 EP disclosed
WO-1999064395-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1999-12-16 WO disclosed
WO-1998053814-A1 HETEROCYCLIC AMIDE COMPOUNDS AS CELL ADHESION INHIBITORS MERCK & CO., INC. (US) 1998-12-03 WO disclosed