SCHEMBL6404056

SCHEMBL6404056

CCC(CCCCCCN)NCc1ccccc1OC

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 13/20 0.58
ATM Q13315 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
GRIN1 Q05586 4/20 0.47
GRIN2A Q12879 4/20 0.47
BCHE P06276 4/20 0.47
ACHE P22303 4/20 0.47
CHRM4 P08173 4/20 0.47
CHRM5 P08912 4/20 0.47
CHRM1 P11229 4/20 0.47
CHRM3 P20309 4/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
TSHR P16473 1/20 0.47
THPO P40225 1/20 0.47
RECQL P46063 1/20 0.47
ALDH1A1 P00352 1/20 0.47
GAA P10253 1/20 0.47
MAPT P10636 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4538523 1.00 CHRM2 (0.58) CHRM2ATML3MBTL1GRIN1GRIN2A
SCHEMBL6313952 0.89 L3MBTL1 (0.54) CHRM2ATML3MBTL1GRIN1GRIN2A
SCHEMBL20988035 0.83 ATM (0.63) CHRM2ATML3MBTL1GRIN1GRIN2A
SCHEMBL5136256 0.82 CHRM2 (0.43) CHRM2ALDH1A1
SCHEMBL6398519 0.81 LMNA (0.43) CHRM2CYP3A4CYP2D6ALDH1A1
SCHEMBL20584486 0.75 CHRM2 (0.80) CHRM2GRIN1GRIN2ABCHEACHE
SCHEMBL4373386 0.75 CHRM2 (0.97) CHRM2GRIN1GRIN2ABCHEACHE
SCHEMBL10288228 0.73 KDM4E (0.40) CHRM2ATML3MBTL1TSHRALDH1A1
SCHEMBL27725768 0.73 CHRM2 (0.54) CHRM2GRIN1GRIN2ABCHEACHE
SCHEMBL29263690 0.72 TAAR1 (0.72) CHRM2ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1497257-A1 2,5-BIS-DIAMINE-[1,4] BENZOQUINONE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE, A PROCESS FOR THEIR PREPARATION AND INTERMEDIATES THEREFOR Alma Mater Studiorum -Universita' di Bologna (IT) 2005-01-19 EP disclosed
WO-2003087035-A1 2,5-BIS-DIAMINE-'1,4! BENZOQUINONE DERIVATIVES FOR THE TREATMENT OF ALZHEIMER'S DISEASE A PROCESS FOR THEIR PREPARATION AND INTERMEDIATES THEREFOR ALMA MATER STUDIORUM-UNIVERSITA' DI BOLOGNA (IT) 2003-10-23 WO disclosed