SCHEMBL6404750

SCHEMBL6404750

FC(F)(F)c1[c]cn(-c2ccccc2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 1/20 0.37
ALDH1A1 P00352 3/20 0.35
MAPT P10636 3/20 0.33
PTGS2 P35354 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
P2RX7 Q99572 1/20 0.33
NOTUM Q6P988 1/20 0.33
POLB P06746 2/20 0.33
HPGD P15428 3/20 0.32
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
ADORA3 P0DMS8 1/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
GAA P10253 1/20 0.32
CASR P41180 1/20 0.31
CYP2C9 P11712 2/20 0.31
MEN1 O00255 1/20 0.31
LMNA P02545 1/20 0.31
CYP1A2 P05177 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23674903 0.84 SRC (0.35) BRAF
SCHEMBL22653988 0.81 ALDH1A1 (0.35) ALDH1A1MAPTPTGS2P2RX7NOTUM
SCHEMBL28777159 0.72 ADORA1 (0.40) ALDH1A1MAPTNPC1RAB9ANOTUM
SCHEMBL1901000 0.71 NPC1 (0.39) ALDH1A1MAPTNPC1RAB9ANOTUM
SCHEMBL1323074 0.69 PTGS2 (0.42) ALDH1A1MAPTPTGS2NPC1RAB9A
SCHEMBL16830498 0.67 ALDH1A1 (0.36) ALDH1A1MAPTNPC1RAB9ANOTUM
SCHEMBL23674906 0.66 HCAR1 (0.35) SMN1; SMN2GAACYP2C9MEN1CYP1A2
SCHEMBL22099773 0.66
SCHEMBL1094013 0.65 NPC1 (0.63) PTGS1ALDH1A1MAPTNPC1RAB9A
SCHEMBL4459050 0.64 PTGS1 (0.41) PTGS1ALDH1A1MAPTPTGS2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050143436-A1 Inhibitors of interleukin-1beta converting enzyme VERTEX PHARMACEUTICALS INCORPORATED 2005-06-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050143436-A1 Inhibitors of interleukin-1beta converting enzyme IL1A, IL1B, IFNAR1 PTGS1 109/4885ALDH1A1 458/4885MAPT 1727/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.