SCHEMBL6414864

SCHEMBL6414864

CCC(C(=O)N1CCC2(CC1)CC(OC(=O)O)=NO2)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
TSHR P16473 4/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
GAA P10253 1/20 0.53
KDM4E B2RXH2 2/20 0.46
LMNA P02545 2/20 0.45
MAPK1 P28482 1/20 0.43
RECQL P46063 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
HSD17B10 Q99714 1/20 0.41
CHRM1 P11229 7/20 0.39
ADORA1 P30542 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
BCHE P06276 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6411364 0.84 ALDH1A1 (0.46) ALDH1A1TSHRL3MBTL1GAAKDM4E
SCHEMBL2400919 0.84 ALDH1A1 (0.59) ALDH1A1TSHRL3MBTL1GAAKDM4E
SCHEMBL15309184 0.77 ALDH1A1 (0.61) ALDH1A1TSHRL3MBTL1GAAKDM4E
SCHEMBL6410215 0.76 SLC6A7 (0.42) ALDH1A1TSHRGAALMNAMAPK1
SCHEMBL2401027 0.75 ALDH1A1 (0.48) ALDH1A1TSHRL3MBTL1GAAKDM4E
SCHEMBL6411469 0.74 RAB9A (0.50) L3MBTL1GAALMNASMN1; SMN2
SCHEMBL4070026 0.73 KDM4E (0.32) KDM4E
SCHEMBL6409811 0.73 TP53 (0.53) ALDH1A1MAPK1
SCHEMBL6418195 0.73 POLB (0.55) ALDH1A1TSHRGAAMAPK1HSD17B10
SCHEMBL6417720 0.72 ALDH1A1 (0.58) ALDH1A1TSHRL3MBTL1MAPK1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1401841-B1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN GRUENENTHAL GMBH (DE) 2005-08-24 EP disclosed
EP-1401841-A1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO 4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN Grünenthal GmbH (DE) 2004-03-31 EP disclosed
WO-2003000699-A1 SUBSTITUTED 1-OXA-2,8-DIAZA-SPIRO[4,5]DEC-2-ENE DERIVATIVES AS MEDICAMENTS FOR THE TREATMENT OF PAIN Grünenthal GmbH (DE) 2003-01-03 WO disclosed