SCHEMBL6419216

SCHEMBL6419216

COc1ccc(C(=CCO)c2ccc(OC)cc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
KDM4E B2RXH2 2/20 0.57
MAPT P10636 2/20 0.57
HPGD P15428 2/20 0.57
NR1I2 O75469 1/20 0.50
SMN1; SMN2 Q16637 2/20 0.48
LMNA P02545 1/20 0.48
ESR1 P03372 1/20 0.48
ADORA3 P0DMS8 1/20 0.48
TSHR P16473 1/20 0.48
MAPK1 P28482 1/20 0.48
CYP2C19 P33261 1/20 0.48
ADRA1A P35348 1/20 0.48
HIF1A Q16665 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HSD17B10 Q99714 1/20 0.48
CES2 O00748 1/20 0.48
CES1 P23141 1/20 0.48
PDE4A P27815 1/20 0.47
PDE4B Q07343 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28062355 0.84 KDM4E (0.53) ALDH1A1KDM4EMAPTHPGDNR1I2
SCHEMBL3952535 0.82 MAPT (0.55) ALDH1A1KDM4EMAPTHPGDNR1I2
SCHEMBL9177747 0.82 KDM4E (0.55) ALDH1A1KDM4EMAPTHPGDNR1I2
SCHEMBL6419828 0.81 L3MBTL1 (0.52) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL6419827 0.81 L3MBTL1 (0.52) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL18897456 0.80 CA1 (0.52) ALDH1A1KDM4EMAPTHPGDNR1I2
SCHEMBL10361923 0.79 KDM4E (0.52) ALDH1A1KDM4EMAPTHPGDNR1I2
SCHEMBL9639091 0.79 CA1 (0.57) ALDH1A1KDM4EMAPTHPGDSMN1; SMN2
SCHEMBL6433983 0.78 CES2 (0.51) ALDH1A1KDM4EMAPTHPGDNR1I2
SCHEMBL6937356 0.78 ALDH1A1 (0.65) ALDH1A1KDM4EMAPTHPGDNR1I2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6972294-B1 Compounds, their preparation and use NOVO NORDISK, A/S (DK) 2005-12-06 US disclosed
EP-1171414-A1 COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2002-01-16 EP disclosed
WO-2000063153-A1 NEW COMPOUNDS, THEIR PREPARATION AND USE NOVO NORDISK A/S (DK) 2000-10-26 WO disclosed