SCHEMBL6422576

SCHEMBL6422576

O=C1CCCC2(CCNCC2)N1Cc1ccccc1-n1nccn1

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 16/20 0.41
HCRTR2 O43614 16/20 0.41
KCNH2 Q12809 1/20 0.38
LTC4S Q16873 1/20 0.38
ROCK2 O75116 2/20 0.34
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2133994 0.77 HCRTR1 (0.53) HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL2135427 0.73 HCRTR1 (0.65) HCRTR1HCRTR2KCNH2LTC4S
SCHEMBL2026638 0.73 HCRTR2 (0.63) HCRTR1HCRTR2
SCHEMBL2023628 0.65 HTR6 (0.62) HCRTR1HCRTR2
SCHEMBL2022006 0.61 TPH1 (0.34) HCRTR1HCRTR2
SCHEMBL5561359 0.60 HTR1A (0.48)
SCHEMBL6111104 0.59 L3MBTL1 (0.51)
SCHEMBL6249596 0.59 L3MBTL1 (0.54)
SCHEMBL2023861 0.58 KDM4E (0.39) HCRTR1HCRTR2
SCHEMBL13543074 0.58 KMT2A (0.48) CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012055888-A1 DIAZA-SPIRO[5.5]UNDECANES USEFUL AS OREXIN RECEPTOR ANTAGONISTS NOVARTIS AG (CH) 2012-05-03 WO disclosed