SCHEMBL6422590

SCHEMBL6422590

O=S(=O)(c1ccccc1)C1CNCCO1

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 11/20 0.38
SLC6A3 Q01959 8/20 0.38
SLC6A4 P31645 6/20 0.38
CYP2D6 P10635 1/20 0.38
KCNH2 Q12809 1/20 0.38
DRD2 P14416 2/20 0.38
HTR2A P28223 2/20 0.38
HTR6 P50406 1/20 0.36
DRD3 P35462 1/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPT P10636 1/20 0.36
ADRB2 P07550 1/20 0.35
HTR1A P08908 1/20 0.35
ADRA1A P35348 1/20 0.35
HTR2B P41595 1/20 0.35
ADRA2C P18825 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28091851 0.85 AKR1C3 (0.47) ALDH1A1MAPT
SCHEMBL10781545 0.84 MAPT (0.44) MAPT
SCHEMBL28433779 0.84 HTR6 (0.39) CYP2D6KCNH2HTR6
SCHEMBL14775611 0.84 HTR6 (0.37) SLC6A2SLC6A4HTR6ALDH1A1
SCHEMBL27828787 0.84 DRD2 (0.40) SLC6A2SLC6A3SLC6A4KCNH2DRD2
SCHEMBL5821011 0.84 MMP2 (0.33) DRD2HTR2ADRD3
SCHEMBL3866888 0.84 DRD2 (0.34) DRD2DRD3HTR1A
SCHEMBL4771959 0.84 GLA (0.35) DRD2DRD3
SCHEMBL16345364 0.83 ENPP2 (0.40) DRD2DRD3
SCHEMBL28285203 0.83 CA12 (0.40) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111440132-B Novel method for preparing oxygen heterocyclic compound by ionic liquid catalysis 中国科学院化学研究所 2022-02-01 CN claimed
CN-111440132-A Novel method for preparing oxygen heterocyclic compound by ionic liquid catalysis 中国科学院化学研究所 2020-07-24 CN claimed
EP-0489085-B1 RIGID-ROD POLYMERS MISSISSIPPI POLYMER TECHNOLOGI (US) 2005-12-07 EP claimed
CN-111440132-B Novel method for preparing oxygen heterocyclic compound by ionic liquid catalysis 中国科学院化学研究所 2022-02-01 CN disclosed
CN-111440132-A Novel method for preparing oxygen heterocyclic compound by ionic liquid catalysis 中国科学院化学研究所 2020-07-24 CN disclosed
CN-110015984-A Substituted (E)-N '-(1- phenylethylene) benzoyl hydrazine analog as histone demethylase inhibitor 犹他大学研究基金会 2019-07-16 CN disclosed
CN-105555784-B Substituted (E) -N' - (1-phenylethylene) benzoyl hydrazine analogs as histone demethylase inhibitors 犹他大学研究基金会 2019-03-15 CN disclosed
CN-105814035-B Bruton's tyrosine kinase inhibitor 豪夫迈·罗氏有限公司 2018-02-02 CN disclosed
US-20170334865-A1 DDR2 INHIBITORS AND METHODS OF USING WASHINGTON UNIVERSITY (US) 2017-11-23 US disclosed
WO-2016070024-A1 DDR2 INHIBITORS AND METHODS OF USING WASHINGTON UNIVERSITY (US) 2016-05-06 WO disclosed
US-20020037888-A1 4-imidazol-1-ylmethyl-2-(2-(2-oxo-piperidin-1-yl)-phenoxy) -benzonitrile for example; farnesyl-protein transferase inhibitors; treating cancer, benign proliferative disorder, hepatitis virus, restenosis, and polycystic kidney disease MERCK & CO., INC. 2002-03-28 US disclosed
US-6284755-B1 Inhibitors of prenyl-protein transferase MERCK & CO., INC. 2001-09-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170334865-A1 DDR2 INHIBITORS AND METHODS OF USING DDR2, DDR1, DDRGK1 SLC6A2 3942/4885SLC6A3 4070/4885SLC6A4 4609/4885
US-20020037888-A1 4-imidazol-1-ylmethyl-2-(2-(2-oxo-piperidin-1-yl)-phenoxy) -benzonitrile for example; farnesyl-protein transferase inhibitors; treating cancer, benign proliferative disorder, hepatitis virus, restenosis, and polycystic kidney disease FNTA, PKD1, FNTB SLC6A2 4798/4885SLC6A3 4559/4885SLC6A4 4401/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.