SCHEMBL6425430

SCHEMBL6425430

O=S(=O)(Cl)c1ccccc1Oc1cc(Cl)cc(Cl)c1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 1/20 0.45
EPAS1 Q99814 15/20 0.41
ACLY P53396 1/20 0.40
LMNA P02545 1/20 0.40
MAPT P10636 1/20 0.40
PGR P06401 1/20 0.38
VEGFA P15692 1/20 0.37
ELANE P08246 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7386055 0.84 TRPV4 (0.46) TRPV4LMNAMAPTPGR
SCHEMBL30307015 0.84 TRPV4 (0.46) TRPV4LMNAMAPTPGR
SCHEMBL997994 0.82 CASP1 (0.48) ACLYLMNAMAPTPGR
SCHEMBL7205989 0.81 TRPV4 (0.42) TRPV4LMNAMAPTPGRELANE
SCHEMBL31387938 0.81 TRPV4 (0.42) TRPV4LMNAMAPTPGRELANE
SCHEMBL4836069 0.80 HTR2A (0.49) TRPV4EPAS1PGR
SCHEMBL5678951 0.80 CASP1 (0.54) TRPV4
SCHEMBL5682872 0.78 GAA (0.53) LMNAMAPT
SCHEMBL8360769 0.77 TSHR (0.41) TRPV4EPAS1LMNAMAPTVEGFA
SCHEMBL926865 0.77 CA12 (0.49) LMNAMAPTELANE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1608374-A1 2-PHENOXY- AND 2-PHENYLSULFOMAMIDE DERIVATIVES WITH CCR3 ANTAGONISTIC ACTIVITY FOR THE TREATMENT OF ASTHMA AND OTHER INFLAMMATORY OR IMMUNOLOGICAL DISORDERS Actimis Pharmaceuticals, Inc. (US) 2005-12-28 EP disclosed
WO-2004084898-A1 2-PHENOXY- AND 2-PHENYLSULFOMAMIDE DERIVATIVES WITH CCR3 ANTAGONISTIC ACTIVITY FOR THE TREATMENT OF ASTHMA AND OTHER INFLAMMATORY OR IMMUNOLOGICAL DISORDERS ACTIMIS PHARMACEUTICALS, INC. (US) 2004-10-07 WO disclosed