SCHEMBL6426953

SCHEMBL6426953

Cn1sc(=O)n(-c2cc(C(C)(C)C)on2)c1=O

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 11/20 0.41
GSK3B P49841 11/20 0.41
HTR7 P34969 1/20 0.39
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
ALOX15 P16050 2/20 0.35
EGFR P00533 2/20 0.34
ALDH1A1 P00352 1/20 0.34
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
CNR1 P21554 1/20 0.30
CNR2 P34972 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10802440 0.77 RGS4 (0.40) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL6428649 0.74 GSK3A (0.53) GSK3AGSK3BMEN1KMT2AALDH1A1
SCHEMBL27260273 0.72 MEN1 (0.39) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL10807029 0.67 HTR7 (0.41) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL8796280 0.66 HTR7 (0.43) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL10961593 0.66 HTR7 (0.43) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL11290248 0.65 ALOX15 (0.35) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL11016128 0.65 HTR7 (0.44) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL11017716 0.65 HTR7 (0.42) HTR7MEN1KMT2AALOX15EGFR
SCHEMBL10991348 0.64 HTR7 (0.41) HTR7MEN1KMT2AALOX15EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005024755-A2 MEDICAMENTS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS OR DIABETES DECIPHERA PHARMACEUTICALS, LLC. (US) 2005-03-17 WO disclosed
EP-0129928-B1 OXAZOLYL-SUBSTITUTED DIAZAHETEROCYCLES SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1987-09-02 EP disclosed
EP-0129928-A1 Oxazolyl-substituted diazaheterocycles SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1985-01-02 EP disclosed
US-4474598-A HERBICIDES SHELL OIL COMPANY (US) 1984-10-02 US disclosed