SCHEMBL6427152

SCHEMBL6427152

CCc1cccc(C(=O)O)c1-c1ccc(C#Cc2ccc(-n3ccnc3)c(C(C)C)c2C)cc1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TBXAS1 P24557 1/20 0.35
DHODH Q02127 1/20 0.31
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
CTSA P10619 1/20 0.31
PDE4A P27815 1/20 0.30
PDE4B Q07343 1/20 0.30
PDE4C Q08493 1/20 0.30
PDE4D Q08499 1/20 0.30
ADH5 P11766 3/20 0.30
ALDH1A1 P00352 1/20 0.30
CYP19A1 P11511 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
FFAR1 O14842 1/20 0.30
AAK1 Q2M2I8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5735868 0.85 ADH5 (0.38) DHODHADH5
SCHEMBL5735900 0.79 FFAR1 (0.40) TBXAS1FFAR1
SCHEMBL6427800 0.78 TDP1 (0.36) ALDH1A1FFAR1AAK1
SCHEMBL7984336 0.74 PDE4A (0.37) TBXAS1DHODHHCRTR1HCRTR2PDE4A
SCHEMBL6427151 0.73 TBXAS1 (0.46) TBXAS1CYP19A1
SCHEMBL5735726 0.70 ADH5 (0.47) TBXAS1ADH5ALDH1A1
SCHEMBL6427628 0.69 TDP1 (0.38) ALDH1A1CYP19A1FFAR1AAK1
SCHEMBL5736507 0.67 FFAR1 (0.44) TBXAS1FFAR1
SCHEMBL5738924 0.66 LMNA (0.49) TBXAS1PDE4APDE4BPDE4CPDE4D
SCHEMBL7980582 0.65 IDO1 (0.49) TBXAS1DHODHADH5ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6369225-B1 ENZYME INHIBITORS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed