SCHEMBL7984336

SCHEMBL7984336

CCc1cc(C#Cc2ccc(-n3ccnc3)c(C)c2C)ccc1C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.37
PDE4B Q07343 2/20 0.37
PDE4C Q08493 2/20 0.37
PDE4D Q08499 2/20 0.37
ADH5 P11766 5/20 0.35
TBXAS1 P24557 1/20 0.34
LMNA P02545 2/20 0.34
STING1 Q86WV6 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
MITF O75030 1/20 0.33
KMT2A Q03164 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
AAK1 Q2M2I8 1/20 0.33
CD274 Q9NZQ7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5735726 0.82 ADH5 (0.47) ADH5TBXAS1ALDH1A1MAPTSMN1; SMN2
SCHEMBL5736507 0.79 FFAR1 (0.44) TBXAS1
SCHEMBL5738924 0.77 LMNA (0.49) PDE4APDE4BPDE4CPDE4DTBXAS1
SCHEMBL6427628 0.76 TDP1 (0.38) LMNAALDH1A1KMT2AAAK1CYP3A4
SCHEMBL6427152 0.74 TBXAS1 (0.35) PDE4APDE4BPDE4CPDE4DADH5
SCHEMBL7984143 0.74 TBXAS1 (0.50) TBXAS1
SCHEMBL5800531 0.72 PDE4A (0.52) PDE4APDE4BPDE4CPDE4DADH5
SCHEMBL15174944 0.70 CSNK2A1 (0.45) PDE4APDE4BPDE4CPDE4DADH5
SCHEMBL5735868 0.69 ADH5 (0.38) ADH5DHODHCYP3A4CYP2D6CYP2C19
SCHEMBL1893489 0.69 MAOB (0.44) PDE4APDE4BPDE4CPDE4DADH5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed