SCHEMBL6427628

SCHEMBL6427628

Cc1c(C#Cc2ccc(C(C)C(=O)O)cc2)ccc(-n2ccnc2)c1C

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.38
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
PTGS2 P35354 5/20 0.33
AAK1 Q2M2I8 1/20 0.32
KMT2A Q03164 1/20 0.32
FFAR1 O14842 3/20 0.32
CD38 P28907 1/20 0.32
MMP9 P14780 1/20 0.32
CYP3A4 P08684 1/20 0.32
BAZ2B Q9UIF8 1/20 0.32
PTGS1 P23219 3/20 0.32
LMNA P02545 2/20 0.32
CYP2C9 P11712 2/20 0.32
AKR1C3 P42330 2/20 0.32
CXCR1 P25024 2/20 0.32
CXCR2 P25025 2/20 0.32
ACACB O00763 1/20 0.32
ALB P02768 1/20 0.32
ESR1 P03372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6427800 0.91 TDP1 (0.36) TDP1ALDH1A1POLBPTGS2AAK1
SCHEMBL5735726 0.84 ADH5 (0.47) ALDH1A1CYP3A4BAZ2BRARB
SCHEMBL5736507 0.81 FFAR1 (0.44) POLBFFAR1
SCHEMBL5738924 0.77 LMNA (0.49) ALDH1A1KMT2ACYP3A4BAZ2BLMNA
SCHEMBL7984336 0.76 PDE4A (0.37) ALDH1A1AAK1KMT2ACYP3A4LMNA
SCHEMBL5735900 0.75 FFAR1 (0.40) FFAR1CYP3A4ACACB
SCHEMBL5735868 0.72 ADH5 (0.38) CYP3A4
SCHEMBL28811546 0.69 IDO1 (0.52) TDP1ALDH1A1KMT2ACYP3A4BAZ2B
SCHEMBL6427152 0.69 TBXAS1 (0.35) ALDH1A1AAK1FFAR1CYP19A1
SCHEMBL17679919 0.66 ADH5 (0.65) ALDH1A1CYP3A4BAZ2BLMNAHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6855512-B2 Methods for identifying inhibitors of cytochrome P450RAI ALLERGAN, INC. (US) 2005-02-15 US disclosed
US-6369261-B1 CYCLOPROPYLBENZENE DERIVATIVE OF ACIDS OR ESTERS ALLERGAN SALES, INC. 2002-04-09 US disclosed
US-6303785-B1 SUBSTITUTED N-CYCLOPROPYLTETRAHYDROISOQUINOLINES ALLERGAN SALES, INC. 2001-10-16 US disclosed