SCHEMBL6432401

SCHEMBL6432401

NC(=S)c1cccc(Cn2c(C(=O)O)c(NC(=S)NCc3ccccc3)c3cc(OCc4ccccc4)ccc32)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F10 P00742 9/20 0.50
PLA2G2A P14555 2/20 0.48
EDNRB P24530 2/20 0.45
EDNRA P25101 2/20 0.45
FOLH1 Q04609 3/20 0.42
F2 P00734 2/20 0.42
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.40
ALDH1A1 P00352 1/20 0.40
POLB P06746 1/20 0.40
ALOX12 P18054 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KLKB1 P03952 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL6436685 0.83 F10 (0.49) F10FOLH1F2RAB9A
SCHEMBL6437281 0.79 F10 (0.48) F10FOLH1F2RAB9A
SCHEMBL6432399 0.75 F10 (0.84) F10F2
Trifluoroacetic Acid SCHEMBL6432605 0.75 F10 (0.50) F10F2
SCHEMBL6432795 0.74 F10 (0.68) F10PLA2G2AF2
SCHEMBL7430298 0.70 F10 (0.83) F10PLA2G2AF2
SCHEMBL6435208 0.69 F10 (0.71) F10EDNRBEDNRAFOLH1F2
SCHEMBL6435201 0.67 F10 (0.81) F10FOLH1F2ALDH1A1
SCHEMBL6432363 0.67 F10 (0.63) F10F2
SCHEMBL8545345 0.67 EDNRB (0.69) PLA2G2AEDNRBEDNRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042287-B1 INDOLE DERIVATIVES AS INHIBITORS OF FACTOR XA AVENTIS PHARMA GMBH (DE) 2005-04-20 EP disclosed
US-6337344-B1 ANTICOAGULANTS AND ENZYME INHIBITORS FOR CARDIOVASCULAR DISORDERS AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 2002-01-08 US disclosed
EP-1042287-A1 INDOLE DERIVATIVES AS INHIBITORS OF FACTOR XA Aventis Pharma Deutschland GmbH (DE) 2000-10-11 EP disclosed
WO-1999033800-A1 INDOLE DERIVATIVES AS INHIBITORS OR FACTOR XA AVENTIS PHARMA DEUTSCHLAND GMBH (DE) 1999-07-08 WO disclosed