SCHEMBL6438849

SCHEMBL6438849

CSc1ccc(-c2[nH]nc(C(=O)CCCO[Si](C)(C)C(C)(C)C)c2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CDC25B P30305 9/20 0.39
MAPT P10636 3/20 0.33
GSK3B P49841 2/20 0.31
PTPN2 P17706 1/20 0.31
PTPN1 P18031 1/20 0.31
PTPN11 Q06124 1/20 0.31
HTT P42858 1/20 0.30
HSD17B10 Q99714 1/20 0.30
DUT P33316 1/20 0.30
LMNA P02545 1/20 0.30
HPGD P15428 1/20 0.30
KMT2A Q03164 1/20 0.30
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3864270 0.92 CDC25B (0.37) CDC25BGSK3BPTPN2PTPN1PTPN11
SCHEMBL5150860 0.88 TRPA1 (0.32)
SCHEMBL6439608 0.74 MAPT (0.45) MAPTGSK3BHSD17B10LMNAHPGD
SCHEMBL3864470 0.73 CHRNA7 (0.49) KMT2ASMN1; SMN2
SCHEMBL6441895 0.71 PKM (0.38) MAPTGSK3BHSD17B10LMNAHPGD
SCHEMBL3864273 0.71 CDC25B (0.35) CDC25BPTPN2PTPN1PTPN11LMNA
SCHEMBL6438007 0.70 PTGS2 (0.45) CDC25B
SCHEMBL8642444 0.67 GSK3B (0.45) MAPTGSK3BHTTHSD17B10LMNA
SCHEMBL5150746 0.65 MDM2 (0.45) KMT2A
SCHEMBL6441497 0.65 ALDH1A1 (0.53) MAPTHSD17B10LMNAHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed