SCHEMBL6441497

SCHEMBL6441497

COC(=O)c1n[nH]c(-c2ccc(SC)cc2)c1-c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.53
LMNA P02545 2/20 0.53
SMN1; SMN2 Q16637 3/20 0.46
KDM4E B2RXH2 4/20 0.44
STAT3 P40763 1/20 0.44
HIF1A Q16665 1/20 0.44
GAA P10253 1/20 0.42
NPC1 O15118 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
CCNE2 O96020 1/20 0.40
CDK4 P11802 1/20 0.40
CCND1 P24385 1/20 0.40
CCNE1 P24864 1/20 0.40
CDK2 P24941 1/20 0.40
RPS6KA3 P51812 1/20 0.40
PTGS2 P35354 1/20 0.40
MAPK1 P28482 2/20 0.39
NPSR1 Q6W5P4 1/20 0.39
HSD17B10 Q99714 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441245 0.89 MAPT (0.45) ALDH1A1LMNASMN1; SMN2KDM4ENPC1
SCHEMBL6439608 0.89 MAPT (0.45) ALDH1A1LMNASMN1; SMN2KDM4ESTAT3
SCHEMBL6440359 0.89 ALDH1A1 (0.41) ALDH1A1LMNASMN1; SMN2KDM4ESTAT3
SCHEMBL6441172 0.89 ALDH1A1 (0.41) ALDH1A1LMNASMN1; SMN2KDM4ESTAT3
SCHEMBL6440017 0.86 TGFBR1 (0.44) ALDH1A1LMNASMN1; SMN2KDM4ESTAT3
SCHEMBL5150566 0.86 ALDH1A1 (0.39) ALDH1A1LMNASMN1; SMN2KDM4ESTAT3
SCHEMBL6444469 0.86 ALDH1A1 (0.41) ALDH1A1LMNASMN1; SMN2KDM4ESTAT3
SCHEMBL5154541 0.81 ALDH1A1 (0.37) ALDH1A1LMNAKDM4EGAANPC1
SCHEMBL6438861 0.76 RPS6KA3 (0.43) ALDH1A1LMNAKDM4EGAANPC1
SCHEMBL28180319 0.76 ALDH1A1 (0.45) ALDH1A1LMNASMN1; SMN2KDM4ESTAT3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed