SCHEMBL6440359

SCHEMBL6440359

COC(=O)c1n[nH]c(-c2ccc(SC)cc2)c1-c1ccc(F)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
LMNA P02545 1/20 0.41
MAPK14 Q16539 6/20 0.39
GCGR P47871 5/20 0.39
MAPK13 O15264 2/20 0.39
ALOX5 P09917 2/20 0.39
MAPK12 P53778 2/20 0.39
MAPK11 Q15759 2/20 0.39
MAP2K4 P45985 1/20 0.39
PRKD3 O94806 1/20 0.39
MAP4K4 O95819 1/20 0.39
LCK P06239 1/20 0.39
RET P07949 1/20 0.39
PRKACA P17612 1/20 0.39
RPS6KB1 P23443 1/20 0.39
MATK P42679 1/20 0.39
FRK P42685 1/20 0.39
MAPK9 P45984 1/20 0.39
CSNK1A1 P48729 1/20 0.39
CSNK1D P48730 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441497 0.89 ALDH1A1 (0.53) ALDH1A1LMNACCNE2CDK4CCND1
SCHEMBL6439608 0.88 MAPT (0.45) ALDH1A1LMNAMAP2K4GSK3BCCNE2
SCHEMBL6441245 0.88 MAPT (0.45) ALDH1A1LMNAGSK3BKDM4ENPC1
SCHEMBL6441172 0.88 ALDH1A1 (0.41) ALDH1A1LMNACCNE2CDK4CCND1
SCHEMBL6444469 0.87 ALDH1A1 (0.41) ALDH1A1LMNAFRKCCNE2CDK4
SCHEMBL5150566 0.85 ALDH1A1 (0.39) ALDH1A1LMNACCNE2CDK4CCND1
SCHEMBL6470454 0.83 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL6440017 0.80 TGFBR1 (0.44) ALDH1A1LMNACCNE2CDK4CCND1
SCHEMBL6623323 0.78 MAPK14 (0.44) MAPK14GCGRMAPK13ALOX5MAPK12
SCHEMBL6622736 0.78 MAPK14 (0.44) MAPK14GCGRMAPK13ALOX5MAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed