SCHEMBL6440587

SCHEMBL6440587

CON(C)C(=O)c1n[nH]c(-c2ccc(SC)cc2)c1-c1ccc(C(F)(F)F)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.36
KDM4E B2RXH2 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ATM Q13315 1/20 0.36
MLYCD O95822 1/20 0.36
BCHE P06276 1/20 0.35
ACHE P22303 1/20 0.35
LIPE Q05469 1/20 0.35
PPARD Q03181 3/20 0.34
PPARG P37231 2/20 0.34
TP53 P04637 1/20 0.33
MAPT P10636 1/20 0.33
PTPN1 P18031 1/20 0.33
NOTUM Q6P988 1/20 0.33
PPARA Q07869 2/20 0.33
IKBKB O14920 1/20 0.32
CCNE2 O96020 1/20 0.32
CDK4 P11802 1/20 0.32
CCND1 P24385 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441895 0.86 PKM (0.38) KDM4ERAB9AACHELIPETP53
SCHEMBL6444469 0.85 ALDH1A1 (0.41) POLBKDM4ENPC1RAB9AATM
SCHEMBL5154541 0.84 ALDH1A1 (0.37) KDM4ENPC1PPARGMAPTCCNE2
SCHEMBL6440359 0.72 ALDH1A1 (0.41) KDM4ENPC1RAB9AMAPTCCNE2
SCHEMBL6441382 0.71 POLB (0.36) POLBKDM4ENPC1RAB9AATM
SCHEMBL6441497 0.71 ALDH1A1 (0.53) KDM4ENPC1RAB9ATP53MAPT
SCHEMBL6439608 0.70 MAPT (0.45) KDM4ENPC1RAB9ATP53MAPT
SCHEMBL6441245 0.70 MAPT (0.45) KDM4ENPC1RAB9ATP53MAPT
SCHEMBL6441172 0.70 ALDH1A1 (0.41) POLBKDM4ENPC1RAB9ATP53
SCHEMBL3869717 0.69 CHRNA7 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1534683-A4 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2005-08-24 EP disclosed
EP-1534683-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-01 EP disclosed
WO-2004002409-A2 CYCLOOXYGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed