SCHEMBL5154541

SCHEMBL5154541

CON(C)C(=O)c1n[nH]c(-c2ccc(SC)cc2)c1-c1ccccc1.C[Al](C)C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.37
LMNA P02545 1/20 0.37
RPS6KA3 P51812 1/20 0.35
PTGS2 P35354 3/20 0.34
CCNE2 O96020 1/20 0.34
CDK4 P11802 1/20 0.34
CCND1 P24385 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
KDM4E B2RXH2 4/20 0.32
MAPT P10636 2/20 0.32
HPGD P15428 3/20 0.32
HSD17B10 Q99714 3/20 0.32
GAA P10253 1/20 0.32
PTGS1 P23219 1/20 0.32
CSNK2A2 P19784 1/20 0.31
KDR P35968 1/20 0.31
CSNK2B P67870 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6441895 0.87 PKM (0.38) ALDH1A1LMNACCNE2CDK4CCND1
SCHEMBL6440587 0.84 POLB (0.36) ALDH1A1CCNE2CDK4CCND1CCNE1
SCHEMBL6441497 0.81 ALDH1A1 (0.53) ALDH1A1LMNARPS6KA3PTGS2CCNE2
SCHEMBL6440359 0.71 ALDH1A1 (0.41) ALDH1A1LMNAPTGS2CCNE2CDK4
SCHEMBL6439608 0.71 MAPT (0.45) ALDH1A1LMNACCNE2CDK4CCND1
SCHEMBL6441172 0.71 ALDH1A1 (0.41) ALDH1A1LMNACCNE2CDK4CCND1
SCHEMBL6441245 0.71 MAPT (0.45) ALDH1A1LMNAKDM4EMAPTHPGD
SCHEMBL6438861 0.70 RPS6KA3 (0.43) ALDH1A1LMNARPS6KA3PTGS2CCNE2
SCHEMBL8640607 0.69 MAPK1 (0.73) ALDH1A1RPS6KA3PTGS2MAPK1NPSR1
SCHEMBL6444469 0.68 ALDH1A1 (0.41) ALDH1A1LMNAPTGS2CCNE2CDK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1539679-A4 OXIME AND/OR HYDRAZONE CONTAINING NITROSATED AND/OR NITROSYLATED CYCLOOXIGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED INC (US) 2007-07-04 EP disclosed
EP-1539679-A2 OXIME AND/OR HYDRAZONE CONTAINING NITROSATED AND/OR NITROSYLATED CYCLOOXIGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE Nitromed, Inc. (US) 2005-06-15 EP disclosed
WO-2004002420-A2 OXIME AND/OR HYDRAZONE CONTAINING NITROSATED AND/OR NITROSYLATED CYCLOOXIGENASE-2 SELECTIVE INHIBITORS, COMPOSITIONS AND METHODS OF USE NITROMED, INC. (US) 2004-01-08 WO disclosed