SCHEMBL6441884

SCHEMBL6441884

CCc1c(C2CC2)nc(N)nc1C1CC1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 3/20 0.40
HRH2 P25021 2/20 0.40
HSD17B10 Q99714 2/20 0.34
USP2 O75604 1/20 0.34
GAA P10253 1/20 0.34
MAPT P10636 1/20 0.34
ALOX15 P16050 1/20 0.34
GFER P55789 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NUDT1 P36639 2/20 0.34
DHFR P00374 4/20 0.34
TLR8 Q9NR97 1/20 0.33
TLR7 Q9NYK1 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
GHSR Q92847 1/20 0.32
CCR2 P41597 3/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
HPGD P15428 1/20 0.31
DRD4 P21917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24979083 0.70 ACHE (0.46) HSD17B10ALOX15ALDH1A1CYP1A2
SCHEMBL30162178 0.70 ACHE (0.46) HSD17B10ALOX15ALDH1A1CYP1A2
SCHEMBL28877816 0.68 DHFR (0.41) HRH3HRH2HSD17B10USP2GAA
SCHEMBL29974011 0.68 DHFR (0.41) HRH3HRH2HSD17B10USP2GAA
SCHEMBL26978231 0.67 CCR2 (0.32) CCR2
SCHEMBL27457600 0.67 PDE10A (0.52) HRH3HRH2HSD17B10USP2GAA
SCHEMBL19174177 0.67 LMNA (0.39) HRH3HRH2HSD17B10USP2GAA
SCHEMBL24978158 0.66 GAA (0.38) HRH3HRH2USP2GAAMAPT
SCHEMBL23264225 0.66 PKM (0.34)
SCHEMBL13653845 0.66 HEXA (0.41) SMN1; SMN2DHFRTLR8TLR7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1499598-A1 CHEMICAL COMPOUNDS WITH DUAL ACTIVITY, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS UCB, S.A. (BE) 2005-01-26 EP disclosed
WO-2003087064-A1 CHEMICAL COMPOUNDS WITH DUAL ACTIVITY, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS UCB, S.A. (BE) 2003-10-23 WO disclosed