SCHEMBL6442565

SCHEMBL6442565

O=CC(Br)c1cc(Br)ccc1OC(F)(F)F

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
ALPL P05186 7/20 0.34
KDR P35968 1/20 0.33
HRH4 Q9H3N8 1/20 0.33
EPHX2 P34913 1/20 0.32
ALDH1A1 P00352 1/20 0.32
MAPK1 P28482 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.31
USP28 Q96RU2 1/20 0.31
USP25 Q9UHP3 1/20 0.31
WDR5 P61964 1/20 0.31
PTGFR P43088 2/20 0.31
SLC6A4 P31645 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28755485 0.83 HRH4 (0.37) MAOAMAOBALPLKDRHRH4
SCHEMBL6445833 0.83 EPAS1 (0.34) ALPLEPHX2
SCHEMBL27643695 0.81 MAOA (0.35) MAOAMAOBALPLKDRHRH4
SCHEMBL5608059 0.79 KCNK3 (0.38) MAOAMAOBALDH1A1L3MBTL1SLC6A4
SCHEMBL3641536 0.79 HTT (0.40) ALDH1A1
SCHEMBL16956764 0.76 MAOA (0.35) MAOAMAOBALPLKDRHRH4
SCHEMBL16952339 0.74 HRH4 (0.39) MAOAMAOBALPLKDRHRH4
SCHEMBL20303638 0.74 HRH4 (0.39) MAOAMAOBALPLKDRHRH4
SCHEMBL6604767 0.74 HRH4 (0.39) MAOAMAOBALPLHRH4SLC6A4
SCHEMBL408055 0.73 PTGDR2 (0.51) MAOAMAOBALPLKDREPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583742-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2005-10-12 EP disclosed
WO-2004060870-A1 NOVEL CB 1 RECEPTOUR INVERSE AGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2004-07-22 WO disclosed