SCHEMBL6442967

SCHEMBL6442967

CN(C#N)C(=O)C(Cc1ccc2ccccc2c1)NC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CTSB P07858 4/20 0.52
CTSS P25774 4/20 0.52
CTSL P07711 3/20 0.52
CTSK P43235 2/20 0.52
MMP9 P14780 2/20 0.50
MMP8 P22894 2/20 0.50
PIN1 Q13526 3/20 0.47
MME P08473 5/20 0.44
ACE P12821 4/20 0.44
CPA1 P15085 2/20 0.44
ACE2 Q9BYF1 2/20 0.44
ITGB1 P05556 1/20 0.43
ITGA4 P13612 1/20 0.43
ITGB7 P26010 1/20 0.43
CTSV O60911 1/20 0.43
CA2 P00918 1/20 0.42
PSMB5 P28074 1/20 0.42
TACR1 P25103 1/20 0.41
PYGL P06737 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6018993 0.90 MMP9 (0.52) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6447376 0.88 ITGB1 (0.48) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6443194 0.88 CTSB (0.51) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6021851 0.87 MMP9 (0.51) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6443832 0.87 CTSL (0.52) CTSBCTSSCTSLCTSKITGB1
SCHEMBL6020300 0.86 CTSL (0.62) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6019856 0.83 MMP9 (0.48) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6019793 0.81 MMP9 (0.54) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6020550 0.81 MMP9 (0.56) CTSBCTSSCTSLCTSKMMP9
SCHEMBL6020748 0.81 CTSB (0.58) CTSBCTSSCTSLCTSKMMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed