SCHEMBL6447376

SCHEMBL6447376

CN(C#N)C(=O)C(Cc1ccccc1)NC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 1/20 0.48
ITGA4 P13612 1/20 0.48
ITGB7 P26010 1/20 0.48
CTSL P07711 5/20 0.48
CTSS P25774 4/20 0.48
CTSK P43235 4/20 0.48
CTSB P07858 3/20 0.48
CHRNB2 P17787 1/20 0.47
CHRNB4 P30926 1/20 0.47
CHRNA3 P32297 1/20 0.47
CHRNA4 P43681 1/20 0.47
CAPN1 P07384 1/20 0.47
TACR2 P21452 1/20 0.46
MMP9 P14780 1/20 0.45
MMP8 P22894 1/20 0.45
MMP14 P50281 1/20 0.45
MEN1 O00255 1/20 0.45
ALDH1A1 P00352 1/20 0.45
KMT2A Q03164 1/20 0.45
CLPP Q16740 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443832 0.93 CTSL (0.52) ITGB1ITGA4ITGB7CTSLCTSS
SCHEMBL6442967 0.88 CTSB (0.52) ITGB1ITGA4ITGB7CTSLCTSS
SCHEMBL6019951 0.88 CTSL (0.50) CTSLCTSSCTSKCTSBMMP9
SCHEMBL6443458 0.86 CTSL (0.47) ITGB1ITGA4ITGB7CTSLCTSS
SCHEMBL6021595 0.86 CTSL (0.50) CTSLCTSSCTSKCTSBMMP9
SCHEMBL6449554 0.84 CTSB (0.45) ITGB1ITGA4ITGB7CTSLCTSS
SCHEMBL5517750 0.84 CTSL (0.64) CTSLCTSSCTSKCTSB
SCHEMBL6021764 0.84 CTSL (0.64) CTSLCTSSCTSKCTSB
SCHEMBL5924629 0.83 CTSB (0.54) ITGB1ITGA4ITGB7CTSLCTSS
SCHEMBL6020939 0.82 CTSL (0.45) CTSLCTSSCTSKCTSBMMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed