SCHEMBL6443832

SCHEMBL6443832

CN(C#N)C(=O)C(Cc1ccc(O)cc1)NC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CTSL P07711 3/20 0.52
CTSB P07858 3/20 0.52
CTSS P25774 3/20 0.52
CTSK P43235 3/20 0.52
ITGB1 P05556 3/20 0.48
ITGA4 P13612 3/20 0.48
ITGB7 P26010 3/20 0.48
CAPN1 P07384 1/20 0.42
TACR2 P21452 1/20 0.41
CLPP Q16740 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447376 0.93 ITGB1 (0.48) CTSLCTSBCTSSCTSKITGB1
SCHEMBL6019617 0.89 CTSL (0.53) CTSLCTSBCTSSCTSKITGB1
SCHEMBL6444324 0.88 CTSL (0.50) CTSLCTSBCTSSCTSKITGB1
SCHEMBL6442967 0.87 CTSB (0.52) CTSLCTSBCTSSCTSKITGB1
SCHEMBL6020053 0.86 CTSL (0.50) CTSLCTSBCTSSCTSK
SCHEMBL6019209 0.85 CTSL (0.67) CTSLCTSBCTSSCTSK
SCHEMBL6021341 0.82 CTSL (0.47) CTSLCTSBCTSSCTSK
SCHEMBL6019951 0.82 CTSL (0.50) CTSLCTSBCTSSCTSK
SCHEMBL6443458 0.81 CTSL (0.47) CTSLCTSBCTSSCTSKITGB1
SCHEMBL6449554 0.81 CTSB (0.45) CTSLCTSBCTSSCTSKITGB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed