SCHEMBL6444957

SCHEMBL6444957

N#CCCNC(=O)C(C(N)=O)c1csc2ccccc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.46
CTSL P07711 1/20 0.39
CTSS P25774 1/20 0.39
CTSK P43235 1/20 0.39
JUN P05412 1/20 0.39
MAPK8 P45983 1/20 0.39
MAPK9 P45984 1/20 0.39
HTR7 P34969 3/20 0.38
HTR1A P08908 2/20 0.38
CMA1 P23946 1/20 0.38
CYP2A6 P11509 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6442426 0.88 ALOX5 (0.51) ALOX5CTSLCTSSCTSKJUN
SCHEMBL6442386 0.78 CTSK (0.42) ALOX5CTSLCTSSCTSKJUN
SCHEMBL6021296 0.78 CTSL (0.38) ALOX5CTSLCTSSCTSKCMA1
SCHEMBL6019645 0.78 DPP4 (0.51) CTSLCTSSCTSKJUNMAPK8
SCHEMBL6449675 0.76 CTSK (0.39) ALOX5CTSLCTSSCTSKJUN
SCHEMBL6447617 0.76 CTSK (0.37) ALOX5CTSLCTSSCTSKJUN
SCHEMBL4308881 0.76 NAMPT (0.44) ALOX5JUNMAPK8MAPK9HDAC1
SCHEMBL6444192 0.76 KDM4E (0.40) ALOX5CTSLCTSSCTSKCMA1
SCHEMBL6446717 0.76 CTSK (0.40) ALOX5CTSLCTSSCTSKCMA1
SCHEMBL6446778 0.75 CNR1 (0.43) CTSLCTSSCTSKPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed