SCHEMBL6446778

SCHEMBL6446778

N#CCCNC(=O)C(C(N)=O)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 4/20 0.43
CNR2 P34972 3/20 0.43
BCAT2 O15382 1/20 0.41
CTSS P25774 5/20 0.40
CTSL P07711 3/20 0.40
CTSB P07858 2/20 0.40
CTSK P43235 3/20 0.39
SRC P12931 1/20 0.39
NR3C2 P08235 1/20 0.39
NAAA Q02083 2/20 0.38
POLB P06746 1/20 0.38
EPHX1 P07099 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6442508 0.87 CNR1 (0.40) CNR1CNR2CTSSCTSLCTSK
SCHEMBL6446787 0.86 CTSS (0.52) CTSSCTSLCTSBCTSK
SCHEMBL6445401 0.84 TNF (0.38) CTSSCTSLCTSBCTSKEPHX1
SCHEMBL14861138 0.78 POLB (0.61) CNR1CNR2POLBEPHX1
SCHEMBL14861481 0.78 HDAC1 (0.56) POLBEPHX1
SCHEMBL7746674 0.77 NAAA (0.60) CNR1CNR2NAAAPOLB
SCHEMBL6444957 0.75 ALOX5 (0.46) CTSSCTSLCTSKPOLB
SCHEMBL6020765 0.75 CTSC (0.59) CTSSCTSK
SCHEMBL6444717 0.74 CTSL (0.47) CNR1CNR2CTSSCTSLCTSB
SCHEMBL6443588 0.73 NPC1 (0.51) CTSSCTSLCTSBCTSKPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed