SCHEMBL6445255

SCHEMBL6445255

CCCCOC(=O)NCC(C(=O)NCCC#N)c1ccc2ccccc2c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
LMNA P02545 1/20 0.44
HPGD P15428 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CYP26A1 O43174 2/20 0.38
CTSS P25774 7/20 0.38
CTSL P07711 4/20 0.38
CTSB P07858 3/20 0.38
CYP2D6 P10635 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
KCNH2 Q12809 1/20 0.37
CTSK P43235 4/20 0.36
CTSD P07339 1/20 0.36
EPHX1 P07099 1/20 0.35
POLB P06746 1/20 0.35
GPR88 Q9GZN0 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6449561 0.96 NPC1 (0.49) NPC1RAB9ASMN1; SMN2LMNACYP26A1
SCHEMBL6442277 0.91 NPC1 (0.49) NPC1RAB9ASMN1; SMN2LMNAHPGD
SCHEMBL6443381 0.90 CYP2D6 (0.40) CTSSCTSLCTSBCYP2D6SLC6A2
SCHEMBL6443774 0.88 NPC1 (0.55) NPC1RAB9ASMN1; SMN2LMNAHPGD
SCHEMBL6443710 0.87 NPC1 (0.54) NPC1RAB9ASMN1; SMN2LMNACYP26A1
SCHEMBL6446829 0.87 CTSS (0.38) NPC1RAB9ASMN1; SMN2CTSSCTSL
SCHEMBL6447648 0.87 MTNR1A (0.40) CTSSCTSLCTSBCYP2D6SLC6A2
SCHEMBL6443928 0.86 CTSK (0.41) LMNACTSSCTSLCTSBCYP2D6
SCHEMBL6445250 0.86 CTSS (0.35) NPC1RAB9ASMN1; SMN2LMNACTSS
SCHEMBL6446503 0.85 SMN1; SMN2 (0.43) NPC1RAB9ASMN1; SMN2LMNAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed