SCHEMBL6447648

SCHEMBL6447648

COC(=O)NCC(C(=O)NCCC#N)c1ccc2ccccc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 3/20 0.40
MTNR1B P49286 2/20 0.40
CTSS P25774 5/20 0.40
CTSK P43235 4/20 0.40
CTSL P07711 3/20 0.40
CYP2D6 P10635 4/20 0.39
CTSB P07858 3/20 0.39
CYP3A4 P08684 2/20 0.39
TSHR P16473 2/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPT P10636 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SLC6A2 P23975 3/20 0.38
SLC6A4 P31645 3/20 0.38
SLC6A3 Q01959 3/20 0.38
ATM Q13315 1/20 0.38
KCNH2 Q12809 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6443381 0.90 CYP2D6 (0.40) MTNR1AMTNR1BCTSSCTSKCTSL
SCHEMBL6444054 0.90 CTSS (0.50) MTNR1AMTNR1BCTSSCTSKCTSL
SCHEMBL6444049 0.89 CTSS (0.50) CTSSCTSKCTSLCTSB
SCHEMBL6446829 0.89 CTSS (0.38) MTNR1AMTNR1BCTSSCTSKCTSL
SCHEMBL6443928 0.89 CTSK (0.41) MTNR1AMTNR1BCTSSCTSKCTSL
SCHEMBL6445255 0.87 NPC1 (0.44) CTSSCTSKCTSLCYP2D6CTSB
SCHEMBL6445366 0.86 CTSS (0.47) CTSSCTSKCTSLCTSBALDH1A1
SCHEMBL6449561 0.85 NPC1 (0.49) CTSSCTSLCTSBTSHR
SCHEMBL6447322 0.84 CTSK (0.42) CTSSCTSKCTSLCTSBATM
SCHEMBL6445250 0.84 CTSS (0.35) MTNR1AMTNR1BCTSSCTSKCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed