SCHEMBL6449561

SCHEMBL6449561

CCCCCCOC(=O)NCC(C(=O)NCCC#N)c1ccc2ccccc2c1

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.49
RAB9A P51151 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
LMNA P02545 1/20 0.47
EPHX1 P07099 1/20 0.39
CYP26A1 O43174 1/20 0.38
TSHR P16473 1/20 0.38
ACHE P22303 6/20 0.37
NAAA Q02083 2/20 0.36
CTSL P07711 1/20 0.36
CTSB P07858 1/20 0.36
CTSS P25774 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445255 0.96 NPC1 (0.44) NPC1RAB9ASMN1; SMN2LMNAEPHX1
SCHEMBL6443710 0.92 NPC1 (0.54) NPC1RAB9ASMN1; SMN2LMNACYP26A1
SCHEMBL6443381 0.88 CYP2D6 (0.40) CTSLCTSBCTSS
SCHEMBL6445531 0.88 NPC1 (0.60) NPC1RAB9ASMN1; SMN2LMNATSHR
SCHEMBL6442277 0.88 NPC1 (0.49) NPC1RAB9ASMN1; SMN2LMNACYP26A1
SCHEMBL6446330 0.85 SMN1; SMN2 (0.48) NPC1RAB9ASMN1; SMN2LMNATSHR
SCHEMBL6446829 0.85 CTSS (0.38) NPC1RAB9ASMN1; SMN2CTSLCTSB
SCHEMBL6447648 0.85 MTNR1A (0.40) TSHRCTSLCTSBCTSS
SCHEMBL6443928 0.85 CTSK (0.41) LMNATSHRCTSLCTSBCTSS
SCHEMBL6443774 0.84 NPC1 (0.55) NPC1RAB9ASMN1; SMN2LMNATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed