SCHEMBL6446288

SCHEMBL6446288

CC(C)COC(=O)NCC(C(=O)NCCC#N)c1csc2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSK P43235 6/20 0.39
CTSS P25774 6/20 0.39
CTSL P07711 5/20 0.39
ALOX5 P09917 1/20 0.38
CTSB P07858 2/20 0.36
ALDH1A1 P00352 2/20 0.36
LMNA P02545 2/20 0.36
NMBR P28336 2/20 0.35
TACR1 P25103 1/20 0.35
CYP2D6 P10635 1/20 0.33
MEN1 O00255 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 1/20 0.33
KAT2A Q92830 1/20 0.32
KAT2B Q92831 1/20 0.32
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
MMP8 P22894 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6445530 0.91 CTSS (0.47) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6446717 0.90 CTSK (0.40) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6449675 0.89 CTSK (0.39) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6442386 0.89 CTSK (0.42) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6450930 0.86 CTSS (0.36) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6443387 0.86 CTSS (0.52) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6449690 0.85 SMN1; SMN2 (0.45) CTSKCTSSCTSLALOX5ALDH1A1
SCHEMBL6446410 0.81 CTSS (0.48) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6448203 0.81 CTSS (0.48) CTSKCTSSCTSLALOX5CTSB
SCHEMBL6021296 0.81 CTSL (0.38) CTSKCTSSCTSLALOX5CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed