SCHEMBL6444047

SCHEMBL6444047

N#CCCNC(=O)C(CNC(=O)c1cccc(C(F)(F)F)c1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSL P07711 5/20 0.53
TACR1 P25103 1/20 0.51
GPR139 Q6DWJ6 1/20 0.51
POLB P06746 3/20 0.49
ALDH1A1 P00352 2/20 0.49
LMNA P02545 1/20 0.46
TP53 P04637 2/20 0.45
TP53BP1 Q12888 1/20 0.45
NPC1 O15118 1/20 0.45
MEN1 O00255 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
KMT2A Q03164 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNK3 O14649 1/20 0.44
NAMPT P43490 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6442129 0.92 CTSL (0.49) CTSLTACR1GPR139POLBALDH1A1
SCHEMBL6446641 0.91 CTSL (0.64) CTSLTACR1GPR139POLBALDH1A1
SCHEMBL6444201 0.89 CTSL (0.47) CTSLTACR1GPR139POLBALDH1A1
SCHEMBL6443588 0.86 NPC1 (0.51) CTSLGPR139POLBNPC1SMN1; SMN2
SCHEMBL6822952 0.84 CTSL (0.61) CTSLTACR1GPR139POLBALDH1A1
SCHEMBL6822574 0.82 CTSL (0.44) CTSLTACR1GPR139POLBALDH1A1
SCHEMBL6444761 0.82 POLB (0.53) CTSLGPR139POLBALDH1A1TP53
SCHEMBL6446599 0.82 GUSB (0.43) CTSLGPR139POLBNPC1SMN1; SMN2
SCHEMBL6822806 0.82 POLB (0.52) CTSLGPR139POLBALDH1A1TP53BP1
SCHEMBL6446794 0.81 CTSL (0.58) CTSLTACR1GPR139POLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed