SCHEMBL6822952

SCHEMBL6822952

N#CCNC(=O)C(CNC(=O)c1cccc(C(F)(F)F)c1)c1ccc(O)cc1

nearest known ligand 0.61

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CTSL P07711 9/20 0.61
ALDH1A1 P00352 1/20 0.49
POLB P06746 1/20 0.49
GPR139 Q6DWJ6 1/20 0.48
NPC1 O15118 1/20 0.47
CTSS P25774 2/20 0.47
CTSK P43235 2/20 0.47
TACR1 P25103 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
TP53BP1 Q12888 1/20 0.45
MAPT P10636 1/20 0.44
TAS1R3 Q7RTX0 1/20 0.44
TAS1R1 Q7RTX1 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446641 0.93 CTSL (0.64) CTSLALDH1A1POLBGPR139NPC1
SCHEMBL6442129 0.90 CTSL (0.49) CTSLALDH1A1POLBGPR139NPC1
SCHEMBL6446794 0.87 CTSL (0.58) CTSLALDH1A1POLBGPR139NPC1
SCHEMBL6443540 0.85 CTSK (0.60) CTSLNPC1CTSSCTSK
SCHEMBL6444047 0.84 CTSL (0.53) CTSLALDH1A1POLBGPR139NPC1
SCHEMBL6822562 0.82 CTSK (0.47) CTSLCTSSCTSK
SCHEMBL6824499 0.81 CTSL (0.62) CTSLALDH1A1POLBGPR139NPC1
SCHEMBL27457044 0.81 POLB (0.68) CTSLALDH1A1POLBGPR139NPSR1
SCHEMBL6446138 0.80 CTSL (0.61) CTSLALDH1A1POLBGPR139NPC1
SCHEMBL6020480 0.79 CTSL (0.84) CTSLCTSSCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO claimed
WO-2004056755-A2 COMPOUNDS FOR THE INHIBITION OF NON-PROTEOLYTIC ENZYMES JERENI AG (DE) 2004-07-08 WO disclosed