SCHEMBL6447225

SCHEMBL6447225

CSC(CNC(=O)OC(C)(C)C)C(=O)NCCC#N

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 16/20 0.44
CTSK P43235 14/20 0.44
CTSL P07711 2/20 0.44
CTSB P07858 2/20 0.44
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6447493 0.87 CTSS (0.57) CTSSCTSKCTSLCTSB
SCHEMBL6446718 0.86 CTSS (0.32) CTSSCTSKCTSLCTSB
SCHEMBL6446773 0.82 ZDHHC20 (0.32)
SCHEMBL1304101 0.81 TDP1 (0.53) CTSSCTSKCTSLCTSBMEN1
SCHEMBL6442039 0.80 SMN1; SMN2 (0.36) CTSSCTSKCTSLCTSB
SCHEMBL6444978 0.79 CTSS (0.42) CTSSCTSKCTSLCTSBMEN1
SCHEMBL6445291 0.78 ACHE (0.42)
SCHEMBL6019683 0.77 CTSS (0.62) CTSSCTSKCTSLCTSB
SCHEMBL15764468 0.77 CTSS (0.62) CTSSCTSKCTSLCTSB
SCHEMBL6445034 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed