SCHEMBL6446718

SCHEMBL6446718

COC(=O)NCC(SC)C(=O)NCCC#N

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CTSS P25774 2/20 0.32
CTSK P43235 2/20 0.32
EPHX1 P07099 1/20 0.31
CTSL P07711 1/20 0.31
CTSB P07858 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6446773 0.87 ZDHHC20 (0.32)
SCHEMBL6447225 0.86 CTSS (0.44) CTSSCTSKCTSLCTSB
SCHEMBL6444153 0.86 CTSS (0.42) CTSSCTSKCTSLCTSB
SCHEMBL6442039 0.85 SMN1; SMN2 (0.36) CTSSCTSKCTSLCTSBMAPT
SCHEMBL6445291 0.83 ACHE (0.42) EPHX1
SCHEMBL6444828 0.81 ACHE (0.47) EPHX1
SCHEMBL6445034 0.81
SCHEMBL6822717 0.79 ALDH1A1 (0.34)
SCHEMBL6447810 0.78 MAPT (0.37) MAPT
SCHEMBL10244410 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed