SCHEMBL6443458

SCHEMBL6443458

CCN(C#N)C(=O)C(Cc1ccccc1)NC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSL P07711 8/20 0.47
CTSS P25774 4/20 0.47
CTSK P43235 4/20 0.47
CTSB P07858 3/20 0.47
CAPN1 P07384 1/20 0.45
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
TACR2 P21452 1/20 0.45
ITGB1 P05556 1/20 0.45
ITGA4 P13612 1/20 0.45
ITGB7 P26010 1/20 0.45
CLPP Q16740 2/20 0.43
SCN1A P35498 1/20 0.41
SCN2A Q99250 1/20 0.41
SCN3A Q9NY46 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6444324 0.94 CTSL (0.50) CTSLCTSSCTSKCTSBCAPN1
SCHEMBL6443194 0.89 CTSB (0.51) CTSLCTSSCTSKCTSBITGB1
SCHEMBL6021087 0.89 CTSL (0.48) CTSLCTSSCTSKCTSBCAPN1
SCHEMBL6019342 0.87 CTSL (0.48) CTSLCTSSCTSKCTSB
SCHEMBL6446903 0.87 CLPP (0.43) CTSBCHRNB2CHRNB4CHRNA3CHRNA4
SCHEMBL6447376 0.86 ITGB1 (0.48) CTSLCTSSCTSKCTSBCAPN1
SCHEMBL6021192 0.85 CTSL (0.62) CTSLCTSSCTSKCTSB
SCHEMBL6445342 0.85 CTSB (0.41) CTSLCTSSCTSKCTSBCHRNB2
SCHEMBL6021771 0.83 LMNA (0.45) CTSLCTSSCTSKCTSB
SCHEMBL6019599 0.83 CTSL (0.52) CTSLCTSSCTSKCTSBCAPN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP claimed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO claimed
EP-1575903-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES Jerini AG (DE) 2005-09-21 EP disclosed
WO-2004065353-A1 COMPOUNDS FOR THE INHIBITION OF ROTAMASES JERINI AG (DE) 2004-08-05 WO disclosed