SCHEMBL6449573

SCHEMBL6449573

COC(=O)n1c(=O)[nH]c(=O)c2ccsc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP15 Q460N3 5/20 0.40
TNKS2 Q9H2K2 5/20 0.40
PARP10 Q53GL7 4/20 0.40
PARP2 Q9UGN5 3/20 0.40
PARP14 Q460N5 1/20 0.40
PARP1 P09874 5/20 0.38
TNKS O95271 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 2/20 0.37
GAA P10253 1/20 0.37
HTT P42858 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
PADI4 Q9UM07 1/20 0.37
ERCC1 P07992 1/20 0.36
ERCC5 P28715 1/20 0.36
FEN1 P39748 1/20 0.36
ERCC4 Q92889 1/20 0.36
SPR P35270 1/20 0.36
KMT2A Q03164 4/20 0.35
MEN1 O00255 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8141804 0.81 PARP1 (0.40) PARP15TNKS2PARP10PARP2PARP14
SCHEMBL2987031 0.74 PARP15 (0.41) PARP15TNKS2PARP10PARP2PARP14
SCHEMBL6674168 0.70 PARP15 (0.41) PARP15TNKS2PARP10PARP2PARP14
SCHEMBL29860930 0.67 CYP1A2 (0.38) ALDH1A1KDM4EGAAHTTNPSR1
SCHEMBL6670689 0.67 ALDH1A1 (0.40) PARP15TNKS2PARP10PARP2ALDH1A1
SCHEMBL19994153 0.64 ERCC1 (0.36) PARP15TNKS2PARP10PARP2PARP1
SCHEMBL10296643 0.64 DAO (0.51) KMT2AMEN1POLB
SCHEMBL31257840 0.63 TNKS2 (0.45) PARP15TNKS2PARP2PARP1TNKS
SCHEMBL27625946 0.62 TYMP (0.55) KMT2AMEN1
SCHEMBL27625945 0.62 SMN1; SMN2 (0.39) ALDH1A1KDM4EGAAHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1536786-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2005-06-08 EP disclosed
WO-2004006913-A1 COMBINATION OF AN ALLOSTERIC INHIBITOR OF MATRIX METALLOPROTEINASE-13 WITH CELECOXIB OR VALDECOXIB WARNER-LAMBERT COMPANY LLC (US) 2004-01-22 WO disclosed