SCHEMBL6457643

SCHEMBL6457643

CCCCCS(=O)(=O)n1ccc2ccc(N3CCCCC3)cc21

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 16/20 0.57
HTR1A P08908 1/20 0.46
DRD2 P14416 1/20 0.46
TERT O14746 1/20 0.37
ADCY5 O95622 1/20 0.36
NPC1 O15118 1/20 0.36
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
NFKB1 P19838 1/20 0.36
RAB9A P51151 1/20 0.36
NFKB2 Q00653 1/20 0.36
KMT2A Q03164 1/20 0.36
RELA Q04206 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1538024 0.74 HTR6 (0.53) HTR6MAPTKMT2AALDH1A1
SCHEMBL7994183 0.69 HTR6 (0.52) HTR6HTR1ADRD2TERTNPC1
SCHEMBL7591875 0.67 HTR6 (0.50) HTR6HTR1ADRD2TERTMAPT
SCHEMBL7034964 0.67 GAA (0.42) HTR6NPC1TP53MAPTNFKB1
SCHEMBL4848922 0.65 CYP2A6 (0.53) HTR6MAPTKMT2AALDH1A1
Hexane SCHEMBL28857999 0.65 DRD2 (0.56) DRD2NPC1TP53MAPTNFKB1
SCHEMBL24220554 0.64 KCNH2 (0.53) DRD2KMT2A
SCHEMBL31743075 0.64 ALDH1A1 (0.49) HTR6HTR1ADRD2TERTMAPT
Hexadecane SCHEMBL28172309 0.64 DRD2 (0.55) DRD2NPC1TP53MAPTNFKB1
SCHEMBL6437205 0.64 HTR6 (0.61) HTR6HTR1ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6897215-B1 Compounds having 5-HT6 receptor antagonist activity NPS ALLELIX CORP. (CA) 2005-05-24 US disclosed
WO-2001032660-A1 COMPOUNDS HAVING 5-HT6 RECEPTOR ANTAGONIST ACTIVITY NPS ALLELIX CORP. (US) 2001-05-10 WO disclosed